SCHEMBL6553742

SCHEMBL6553742

CC(C)(C)OC(=O)C(C)(C)Sc1ccc(CCNC(=O)Cc2ccccc2N2CCOCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
TAAR1 Q96RJ0 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GAA P10253 1/20 0.39
POLB P06746 2/20 0.39
RAB9A P51151 1/20 0.39
AKT1 P31749 1/20 0.39
MAPT P10636 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
PTPN1 P18031 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6552237 0.70 STS (0.53) MEN1KMT2APOLBRAB9AMAPT
SCHEMBL3706363 0.69 NAMPT (0.52) ALDH1A1MEN1KMT2AAKT1MAPT
SCHEMBL11303063 0.69 GAA (0.53) ALDH1A1TAAR1MEN1KMT2AGAA
SCHEMBL6129053 0.69 PPARA (0.47) ALDH1A1MEN1KMT2APOLBRAB9A
SCHEMBL6553673 0.68 PPARA (0.59) ALDH1A1KMT2AGAAPOLBRAB9A
SCHEMBL6774346 0.68 CA12 (0.48) ALDH1A1MEN1KMT2APOLBRAB9A
SCHEMBL7871514 0.66 KMT2A (0.47) KMT2AAKT1
SCHEMBL3884314 0.66 TAAR1 (0.38) ALDH1A1TAAR1KMT2ACYP1A2CYP2C19
SCHEMBL3885465 0.65 CASP3 (0.45) ALDH1A1TAAR1MEN1KMT2AGAA
SCHEMBL6554165 0.64 ALDH1A1 (0.55) ALDH1A1MEN1KMT2AGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1149063-B1 UREIDO-THIOBUTYRIC ACID DERIVATIVES AS PPAR-AGONISTS SMITHKLINE BEECHAM CORP (US) 2004-12-15 EP disclosed
EP-1149063-A2 UREIDO-THIOBUTYRIC ACID DERIVATIVES AS PPAR-AGONISTS GLAXO GROUP LIMITED (GB) 2001-10-31 EP disclosed
US-6306854-B1 ARYLTHIOALKYLACIDS AND ALKYL UREAS GLAXOSMITHKLINE 2001-10-23 US disclosed
WO-2000023407-A2 UREIDO-THIOBUTYRIC ACID DERIVATIVES AS PPAR-AGONISTS GLAXO GROUP LIMITED (GB) 2000-04-27 WO disclosed