SCHEMBL6557623

SCHEMBL6557623

CC(C)(NC(=O)C(C(N)=O)S(=O)(=O)Cc1ccccc1)C(O)C(=O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.38
PRSS1 P07477 3/20 0.35
F2 P00734 2/20 0.35
PRSS2 P07478 2/20 0.35
PRSS3 P35030 2/20 0.35
MDM2 Q00987 1/20 0.35
HPGD P15428 1/20 0.34
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
CTSL P07711 1/20 0.34
CA1 P00915 3/20 0.33
CA2 P00918 3/20 0.33
CA9 Q16790 2/20 0.33
VNN1 O95497 1/20 0.33
CA12 O43570 1/20 0.33
CTSG P08311 1/20 0.33
CTRB1 P17538 1/20 0.33
CMA1 P23946 1/20 0.33
MMP1 P03956 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5445816 0.81 HPGD (0.40) KMT2AMDM2HPGDSLC1A3SLC1A2
SCHEMBL7551628 0.71 CTSS (0.49) CTSL
SCHEMBL5445806 0.69 ALDH1A1 (0.34) KMT2APRSS1F2PRSS2PRSS3
SCHEMBL6557583 0.67 SLC1A3 (0.37) PRSS1F2PRSS2PRSS3SLC1A3
SCHEMBL6560207 0.66 GRM7 (0.37) PRSS1F2PRSS2PRSS3SLC1A3
SCHEMBL6062861 0.65 PRSS1 (0.49) KMT2APRSS1F2PRSS2PRSS3
SCHEMBL7256952 0.65 PRSS1 (0.49) KMT2APRSS1F2PRSS2PRSS3
SCHEMBL6559792 0.64 USP2 (0.39) PRSS1F2HPGDSLC1A3SLC1A2
SCHEMBL10444753 0.64 CES1 (0.52) MDM2KDM4EALDH1A1TSHRHSD17B10
SCHEMBL6557593 0.64 KEAP1 (0.41) MMP1MMP2MMP9MMP8MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1436255-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS Aventis Pharmaceuticals, Inc. (US) 2004-07-14 EP claimed
WO-2003024924-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2003-03-27 WO claimed