SCHEMBL6559792

SCHEMBL6559792

NC(=O)[C@H](C(=O)NC1C(O)CCCC1O)S(=O)(=O)Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 1/20 0.39
F2 P00734 4/20 0.37
F10 P00742 3/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
CA5A P35218 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
CA13 Q8N1Q1 1/20 0.37
CA14 Q9ULX7 1/20 0.37
CA5B Q9Y2D0 1/20 0.37
ALDH1A1 P00352 2/20 0.37
CCR4 P51679 1/20 0.36
MME P08473 1/20 0.36
ACE P12821 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557583 0.84 SLC1A3 (0.37) F2CA12CA1CA2CA4
SCHEMBL6557913 0.81 GBA1 (0.39) F2F10CA12CA1CA2
SCHEMBL5447012 0.80 ALDH1A1 (0.38) USP2HPGDHSD17B10F2ALDH1A1
SCHEMBL6560207 0.78 GRM7 (0.37) F2CA12CA1CA2CA4
SCHEMBL7551628 0.70 CTSS (0.49)
SCHEMBL6558896 0.68 CYP3A4 (0.37) F2CA1CA2CA5ACA9
SCHEMBL6848129 0.68 CTSS (0.53)
SCHEMBL6557593 0.65 KEAP1 (0.41) ALDH1A1
SCHEMBL6557623 0.64 KMT2A (0.38) HPGDHSD17B10F2CA12CA1
SCHEMBL6062861 0.63 PRSS1 (0.49) HPGDHSD17B10F2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1436255-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS Aventis Pharmaceuticals, Inc. (US) 2004-07-14 EP disclosed
WO-2003024924-A1 NOVEL COMPOUNDS AND COMPOSITIONS AS CATHEPSIN INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2003-03-27 WO disclosed