SCHEMBL6558448

SCHEMBL6558448

CC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)NC(C)C(=O)C(F)(F)F)C(C)C)C(C)C

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PSENEN Q9NZ42 1/20 0.39
CASP1 P29466 2/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.32
SIRT5 Q9NXA8 1/20 0.32
CTSD P07339 2/20 0.32
ELANE P08246 2/20 0.32
CASP3 P42574 1/20 0.31
HTRA1 Q92743 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6559665 0.89 PSENEN (0.43) PSENENCASP1CTSDELANE
SCHEMBL6559645 0.88 ALDH1A1 (0.40) PSENENFNTAFNTBCTSD
SCHEMBL6558875 0.87 CASP1 (0.42) PSENENCASP1CTSDCASP3
SCHEMBL6558747 0.86 BACE1 (0.42) PSENENCASP1CTSD
SCHEMBL6560709 0.86 PSENEN (0.41) PSENENCASP1CTSDELANE
SCHEMBL6558465 0.86 PSENEN (0.41) PSENENCASP1CTSDELANE
SCHEMBL6558450 0.84 MAGI3 (0.37) PSENENCASP1CTSDCASP3
SCHEMBL6558839 0.84 PSENEN (0.36) PSENENCASP1CTSDELANECASP3
SCHEMBL6558811 0.83 FURIN (0.46)
SCHEMBL6558805 0.81 HTRA1 (0.47) HTRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948523-B1 PEPTIDOMIMETIC INHIBITORS OF THE HUMAN CYTOMEGALOVIRUS PROTEASE BOEHRINGER INGELHEIM CA LTD (CA) 2004-03-17 EP claimed
US-6291640-B1 OLIGOPEPTIDES; SOLID PHASE SYNTHESIS BOEHRINGER INGELHEIM LTD. (CA) 2001-09-18 US claimed
EP-0948523-B1 PEPTIDOMIMETIC INHIBITORS OF THE HUMAN CYTOMEGALOVIRUS PROTEASE BOEHRINGER INGELHEIM CA LTD (CA) 2004-03-17 EP disclosed
US-6291640-B1 OLIGOPEPTIDES; SOLID PHASE SYNTHESIS BOEHRINGER INGELHEIM LTD. (CA) 2001-09-18 US disclosed