SCHEMBL6558805

SCHEMBL6558805

CC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](Cc1ccccc1)C(=O)NC(C)C(=O)C(F)(F)F)C(C)C)C(C)C

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTRA1 Q92743 10/20 0.47
BACE1 P56817 1/20 0.47
GNPAT O15228 1/20 0.47
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23600925 0.84 ACE (0.55) BACE1GNPATCTSSCTSK
SCHEMBL23572632 0.84 ACE (0.55) BACE1GNPATCTSSCTSK
SCHEMBL23572631 0.84 ACE (0.55) BACE1GNPATCTSSCTSK
SCHEMBL7270319 0.82 CTSS (0.52) GNPATCTSSCTSK
SCHEMBL6558875 0.81 CASP1 (0.42) BACE1GNPAT
SCHEMBL6558448 0.81 PSENEN (0.39) HTRA1
SCHEMBL29112224 0.81 MME (0.58) BACE1GNPAT
SCHEMBL6559665 0.80 PSENEN (0.43)
SCHEMBL6559645 0.80 ALDH1A1 (0.40)
SCHEMBL23600939 0.80 CTSD (0.55) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948523-B1 PEPTIDOMIMETIC INHIBITORS OF THE HUMAN CYTOMEGALOVIRUS PROTEASE BOEHRINGER INGELHEIM CA LTD (CA) 2004-03-17 EP claimed
US-6291640-B1 OLIGOPEPTIDES; SOLID PHASE SYNTHESIS BOEHRINGER INGELHEIM LTD. (CA) 2001-09-18 US claimed
EP-0948523-B1 PEPTIDOMIMETIC INHIBITORS OF THE HUMAN CYTOMEGALOVIRUS PROTEASE BOEHRINGER INGELHEIM CA LTD (CA) 2004-03-17 EP disclosed
US-6291640-B1 OLIGOPEPTIDES; SOLID PHASE SYNTHESIS BOEHRINGER INGELHEIM LTD. (CA) 2001-09-18 US disclosed