SCHEMBL6561886

SCHEMBL6561886

CN(C(=O)c1ccc(C#CCNc2ccc(C(=N)N)cc2)cc1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.53
ACACB O00763 2/20 0.49
HTT P42858 1/20 0.48
SIRT2 Q8IXJ6 1/20 0.47
KMT2A Q03164 2/20 0.44
NPC1 O15118 1/20 0.44
PKM P14618 1/20 0.44
RAB9A P51151 1/20 0.44
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MAOA P21397 1/20 0.42
F2 P00734 3/20 0.40
ALDH1A1 P00352 1/20 0.40
NR1H3 Q13133 1/20 0.40
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
MRGPRX1 Q96LB2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563743 0.87 PRSS1 (0.43) ACACBF2
SCHEMBL6563594 0.86 KMT2A (0.51) ACACBHTTSIRT2KMT2ANPC1
SCHEMBL6563625 0.84 PRSS1 (0.43) PKMRAB9AF2ALDH1A1MRGPRX1
SCHEMBL6565690 0.84 PLAU (0.54) PLAUHTTSIRT2KMT2ANPC1
SCHEMBL6563250 0.84 PLAU (0.54) PLAUACACBHTTSIRT2KMT2A
SCHEMBL6563677 0.83 MRGPRX1 (0.43) ACACBF2MRGPRX1
SCHEMBL6565956 0.82 PLAU (0.49) PLAUACACBHTTSIRT2KMT2A
SCHEMBL6563734 0.82 LTB4R2 (0.45) ACACBKMT2ANPC1F2ALDH1A1
SCHEMBL6563749 0.82 ITGB3 (0.41) ACACBF2ITGB3ITGA2B
SCHEMBL6561827 0.80 MRGPRX1 (0.51) F2MRGPRX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed