SCHEMBL6562437

SCHEMBL6562437

Cc1nc2ccccc2n1Cc1cccc(C#CCNc2ccc(C(=N)N)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 2/20 0.47
KLK1 P06870 1/20 0.47
TNF P01375 1/20 0.46
HDAC1 Q13547 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
GALR3 O60755 2/20 0.42
NR2F2 P24468 2/20 0.42
RAB9A P51151 2/20 0.42
MAPT P10636 5/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
PKM P14618 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
TSHR P16473 2/20 0.41
TP53 P04637 2/20 0.41
NPC1 O15118 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6562124 0.80 KLK5 (0.47) KLK5KLK1ALDH1A1TSHRTP53
SCHEMBL4320699 0.76 KLK1 (0.71) KLK5KLK1RAB9AMAPTKDM4E
SCHEMBL30583224 0.76 KLK1 (0.71) KLK5KLK1RAB9AMAPTKDM4E
Hydrochloric Acid SCHEMBL7408509 0.76 KLK1 (0.70) KLK5KLK1RAB9AMAPTKDM4E
SCHEMBL6563255 0.75 PRSS1 (0.44) KLK5KLK1F10
SCHEMBL21067963 0.73 HDAC1 (0.44) KLK5KLK1TNFHDAC1HDAC6
SCHEMBL7673744 0.72 ASIC3 (0.40) KLK5KLK1F10
SCHEMBL12589583 0.70 F2 (0.55) KLK5KLK1TNFHDAC1HDAC6
SCHEMBL6561827 0.70 MRGPRX1 (0.51) F10
SCHEMBL15567678 0.69 TNF (0.70) TNFHDAC1HDAC6GALR3NR2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed