SCHEMBL6562742

SCHEMBL6562742

CC(=O)Oc1ccccc1C(=O)c1cccc2c1C(=O)NC2=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
HSD17B10 Q99714 3/20 0.49
ALDH1A1 P00352 3/20 0.49
HPGD P15428 3/20 0.49
PTGS2 P35354 2/20 0.49
ESR1 P03372 1/20 0.49
ITGB3 P05106 1/20 0.49
ITGA2B P08514 1/20 0.49
HMGB1 P09429 1/20 0.49
TSHR P16473 1/20 0.49
GGT1 P19440 1/20 0.49
PTGS1 P23219 1/20 0.49
BLM P54132 1/20 0.49
NAPRT Q6XQN6 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
LMNA P02545 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CASP3 P42574 6/20 0.47
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6634972 0.84 KDM4E (0.54) KDM4EHSD17B10ALDH1A1HPGDPTGS2
SCHEMBL22033199 0.81 CASP3 (0.69) KDM4EHSD17B10ALDH1A1HPGDCASP3
SCHEMBL189443 0.79 PTGS2 (0.74) KDM4EHSD17B10ALDH1A1HPGDPTGS2
SCHEMBL30641073 0.79 KMT2A (0.51) KDM4EHSD17B10ALDH1A1HPGDCYP2C9
SCHEMBL9686151 0.78 CASP3 (0.51) KDM4EHSD17B10ALDH1A1HPGDTDP1
SCHEMBL11612938 0.78 KDM4E (0.49) KDM4EHSD17B10ALDH1A1HPGDCASP3
Diphenylether SCHEMBL3762390 0.77 MAOA (0.50) KDM4EHSD17B10ALDH1A1HPGDCASP3
SCHEMBL5128860 0.76 KDM4E (0.58) KDM4EHSD17B10ALDH1A1HPGDCASP3
SCHEMBL8094145 0.74 KDM4E (0.47) KDM4EHSD17B10ALDH1A1HPGDPTGS2
SCHEMBL8094143 0.74 KDM4E (0.47) KDM4EHSD17B10ALDH1A1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817643-A4 COMPOUNDS AND COMPOSITIONS FOR DELIVERING ACTIVE AGENTS EMISPHERE TECH INC (US) 2004-10-06 EP disclosed
EP-0817643-A1 COMPOUNDS AND COMPOSITIONS FOR DELIVERING ACTIVE AGENTS Emisphere Technologies, Inc. (US) 1998-01-14 EP disclosed