SCHEMBL6563536

SCHEMBL6563536

CC(C)(C)OC(=O)NC(=N)c1ccc(NCC#Cc2ccc(C(=O)c3ccccc3)s2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 7/20 0.39
PPARA Q07869 7/20 0.39
PPARD Q03181 2/20 0.39
PTPN11 Q06124 1/20 0.36
HPGD P15428 3/20 0.34
ADRA2C P18825 1/20 0.34
MAOA P21397 1/20 0.34
ADRA1A P35348 1/20 0.34
DRD3 P35462 1/20 0.34
KCNH2 Q12809 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 3/20 0.33
ALDH1A1 P00352 2/20 0.33
PTPRB P23467 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563256 0.81 HPGD (0.45) HPGDADRA2CMAOAADRA1ADRD3
SCHEMBL7673754 0.81 NQO2 (0.41) HPGDADRA2CMAOAADRA1ADRD3
SCHEMBL6563729 0.80 PPARG (0.41) PPARGPPARAPPARDPTPN11PTPRB
SCHEMBL6563355 0.78 PTPN11 (0.47) PPARGPPARAPPARDPTPN11CTSK
SCHEMBL6565434 0.77 PTPN11 (0.41) PPARGPPARAPPARDPTPN11KMT2A
SCHEMBL6563676 0.76 NAMPT (0.42) PPARGPPARAPPARDPTPN11CYP3A4
SCHEMBL6563070 0.76 PTPN11 (0.44) PPARGPPARAPPARDPTPN11KMT2A
SCHEMBL7158402 0.74 PPARG (0.47) PPARGPPARAPPARDKMT2AALDH1A1
SCHEMBL6563323 0.73 MAPT (0.38) PPARGPPARAPPARDPTPN11MAPT
SCHEMBL6563283 0.73 PTPN11 (0.46) PTPN11HPGDALDH1A1MAPTPTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed