SCHEMBL6561835

SCHEMBL6561835

CC1CCCN1C(=O)c1ccc(C#CCNc2ccc(C(=N)NC(=O)OC(C)(C)C)cc2)cc1CO

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.35
HRH3 Q9Y5N1 4/20 0.34
HSD11B1 P28845 1/20 0.34
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
NAMPT P43490 1/20 0.33
HTT P42858 1/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 3/20 0.32
HPGD P15428 2/20 0.32
ACHE P22303 1/20 0.32
BACE1 P56817 1/20 0.32
ALDH1A1 P00352 2/20 0.32
KCNK3 O14649 2/20 0.32
MAPT P10636 1/20 0.32
CMA1 P23946 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565417 0.92 PTPN11 (0.36) PTPN11HRH3HSD11B1DDB1CRBN
SCHEMBL6563002 0.88 HRH3 (0.42) PTPN11HRH3HSD11B1NAMPTNPC1
SCHEMBL6561843 0.87 GAA (0.31) PTPN11HRH3HSD11B1DDB1CRBN
SCHEMBL6563261 0.85 HSD11B1 (0.38) HRH3HSD11B1NAMPTHTTGAA
SCHEMBL6563752 0.84 GAA (0.35) HRH3HSD11B1NAMPTHTTNPC1
SCHEMBL6563591 0.82 LRRK2 (0.39) HRH3HSD11B1NAMPTHTTGAA
SCHEMBL6563605 0.82 GAA (0.37) HRH3HSD11B1NAMPTHTTNPC1
SCHEMBL6563511 0.80 PTPN11 (0.40) PTPN11HSD11B1NPC1
SCHEMBL6563779 0.80 KCNK3 (0.38) PTPN11HSD11B1GAAKCNK3MEN1
SCHEMBL6565533 0.80 ACACB (0.45) PTPN11HSD11B1DDB1CRBNGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed