SCHEMBL6565257

SCHEMBL6565257

CC(=O)c1nc2c(Oc3ccccc3)cccc2cc1O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TTR P02766 2/20 0.41
TSPO P30536 1/20 0.40
P2RX3 P56373 2/20 0.39
MIF P14174 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
EGLN1 Q9GZT9 2/20 0.38
CTNNB1 P35222 1/20 0.38
POLB P06746 1/20 0.38
HSD17B14 Q9BPX1 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6564114 0.88 POLB (0.45) KDM4EHSD17B10POLBMEN1KMT2A
SCHEMBL6566232 0.84 MAPT (0.48) KDM4EKMT2A
SCHEMBL6567173 0.83 LMNA (0.49) KDM4EHSD17B10POLBMEN1KMT2A
SCHEMBL6565243 0.80 MCHR1 (0.48) KDM4EPOLBMEN1KMT2A
SCHEMBL6565264 0.76 MCHR1 (0.51) MEN1KMT2A
SCHEMBL6567192 0.74 MCHR1 (0.53) MEN1KMT2A
SCHEMBL6565253 0.74 TDP1 (0.43) EGLN1KMT2A
SCHEMBL6565245 0.74 DAO (0.41) KDM4EHSD17B10MEN1KMT2A
SCHEMBL6564103 0.74 MAOB (0.48) KDM4EMEN1KMT2A
SCHEMBL2975427 0.70 KDM4E (0.56) KDM4EHSD17B14MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765871-B1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors FIBROGEN INC (US) 2004-03-31 EP disclosed
EP-0765871-A1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-02 EP disclosed