SCHEMBL6565446

SCHEMBL6565446

N#CN(C(=O)C(COC(=O)NCc1ccccc1)C1CC1)C1CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 1/20 0.40
CASP1 P29466 1/20 0.38
BCHE P06276 2/20 0.37
CTSL P07711 4/20 0.36
CTSB P07858 4/20 0.36
CTSS P25774 4/20 0.36
CTSK P43235 4/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36
CCNK O75909 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CDK12 Q9NYV4 1/20 0.36
PLAU P00749 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565489 0.81 CTSS (0.47) MCL1CTSLCTSBCTSSCTSK
SCHEMBL6565444 0.77 CTSL (0.42) MCL1BCHECTSLCTSBCTSS
SCHEMBL6565044 0.76 CHRNB2 (0.41) CASP1CTSLCTSBCTSSCTSK
SCHEMBL6565039 0.76 CTSS (0.46) MCL1CTSLCTSBCTSSCTSK
SCHEMBL6565436 0.74 CTSL (0.39) CASP1BCHECTSLCTSSALDH1A1
SCHEMBL6567346 0.73 L3MBTL1 (0.40) MCL1CTSLCTSBCTSSCTSK
SCHEMBL7438096 0.71 CTSS (0.42) CASP1CTSLCTSBCTSSCTSK
SCHEMBL3899355 0.70 HPGD (0.42) MCL1BCHECTSLCTSBCTSS
SCHEMBL6563724 0.70 CTSS (0.48) CTSLCTSBCTSSCTSK
SCHEMBL6563875 0.69 CTSS (0.50) CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed