SCHEMBL6565444

SCHEMBL6565444

N#CN(C(=O)C(CC1CC1)OC(=O)NCc1ccccc1)C1CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 4/20 0.42
CTSB P07858 4/20 0.42
CTSK P43235 4/20 0.42
CTSS P25774 3/20 0.42
MCL1 Q07820 1/20 0.40
BCHE P06276 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
UTS2R Q9UKP6 1/20 0.36
KLK7 P49862 1/20 0.36
CCNK O75909 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CDK12 Q9NYV4 1/20 0.36
CCR5 P51681 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3902637 0.87 CTSL (0.48) CTSLCTSBCTSKCTSSMCL1
SCHEMBL6565039 0.86 CTSS (0.46) CTSLCTSBCTSKCTSSMCL1
SCHEMBL6565429 0.82 CTSL (0.40) CTSLCTSBCTSKCTSSMCL1
SCHEMBL6567343 0.81 UTS2R (0.42) CTSLCTSBCTSKCTSSALDH1A1
SCHEMBL3902634 0.80 CTSS (0.49) CTSLCTSBCTSKCTSSMCL1
SCHEMBL3893070 0.77 CTSS (0.43) CTSLCTSBCTSKCTSSUTS2R
SCHEMBL3893067 0.77 CTSK (0.43) CTSLCTSBCTSKCTSSHPGD
SCHEMBL6565446 0.77 MCL1 (0.40) CTSLCTSBCTSKCTSSMCL1
SCHEMBL3898975 0.76 CTSS (0.53) CTSLCTSBCTSS
SCHEMBL3910486 0.76 CTSL (0.46) CTSLCTSBCTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed