SCHEMBL6565455

SCHEMBL6565455

CC(C)CC(OC(=O)NCc1ccccc1)C(=O)N(C#N)CCCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.45
CTSL P07711 4/20 0.45
CTSB P07858 4/20 0.45
CTSK P43235 4/20 0.45
UTS2R Q9UKP6 1/20 0.41
MMP8 P22894 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
HPGD P15428 1/20 0.38
ANPEP P15144 1/20 0.38
EPHX2 P34913 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6567349 0.90 CTSS (0.47) CTSSCTSLCTSBCTSKUTS2R
SCHEMBL6565429 0.84 CTSL (0.40) CTSSCTSLCTSBCTSKUTS2R
SCHEMBL3894952 0.84 CTSL (0.54) CTSSCTSLCTSBCTSKUTS2R
SCHEMBL3894949 0.79 CTSS (0.56) CTSSCTSLCTSBCTSKANPEP
SCHEMBL6565039 0.78 CTSS (0.46) CTSSCTSLCTSBCTSKUTS2R
SCHEMBL6567343 0.77 UTS2R (0.42) CTSSCTSLCTSBCTSKUTS2R
SCHEMBL3899392 0.76 CTSL (0.50) CTSSCTSLCTSBCTSKMMP8
SCHEMBL7310650 0.76 ALDH1A1 (0.51) MMP8PPARGPPARAANPEPMEN1
SCHEMBL3907700 0.75 CTSS (0.46) CTSSCTSLCTSBCTSKUTS2R
SCHEMBL3895384 0.75 CTSC (0.55) CTSSCTSLCTSBCTSKPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed