SCHEMBL6567343

SCHEMBL6567343

CC(C)CCN(C#N)C(=O)C(CC1CC1)OC(=O)NCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
UTS2R Q9UKP6 1/20 0.42
CTSL P07711 6/20 0.41
CTSB P07858 6/20 0.41
CTSK P43235 6/20 0.41
CTSS P25774 5/20 0.41
L3MBTL1 Q9Y468 1/20 0.39
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
CASP3 P42574 1/20 0.35
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
CCR5 P51681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6565429 0.87 CTSL (0.40) UTS2RCTSLCTSBCTSKCTSS
SCHEMBL6567349 0.87 CTSS (0.47) UTS2RCTSLCTSBCTSKCTSS
SCHEMBL3902637 0.85 CTSL (0.48) UTS2RCTSLCTSBCTSKCTSS
SCHEMBL6565444 0.81 CTSL (0.42) UTS2RCTSLCTSBCTSKCTSS
SCHEMBL3902634 0.78 CTSS (0.49) CTSLCTSBCTSKCTSS
SCHEMBL6565455 0.77 CTSS (0.45) UTS2RCTSLCTSBCTSKCTSS
SCHEMBL3906527 0.77 CTSL (0.45) CTSLCTSBCTSKCTSSCASP3
SCHEMBL3893070 0.75 CTSS (0.43) UTS2RCTSLCTSBCTSKCTSS
SCHEMBL3893067 0.75 CTSK (0.43) UTS2RCTSLCTSBCTSKCTSS
SCHEMBL6565039 0.74 CTSS (0.46) UTS2RCTSLCTSBCTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed