SCHEMBL6565429

SCHEMBL6565429

N#CN(CCCc1ccccc1)C(=O)C(CC1CC1)OC(=O)NCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.40
CTSB P07858 3/20 0.40
CTSS P25774 3/20 0.40
CTSK P43235 2/20 0.40
UTS2R Q9UKP6 1/20 0.38
BCHE P06276 2/20 0.37
EPHX2 P34913 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
LMNA P02545 1/20 0.35
MMP1 P03956 2/20 0.35
MMP2 P08253 2/20 0.35
MMP3 P08254 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MCL1 Q07820 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6567343 0.87 UTS2R (0.42) CTSLCTSBCTSSCTSKUTS2R
SCHEMBL6565455 0.84 CTSS (0.45) CTSLCTSBCTSSCTSKUTS2R
SCHEMBL3902637 0.83 CTSL (0.48) CTSLCTSBCTSSCTSKUTS2R
SCHEMBL6565444 0.82 CTSL (0.42) CTSLCTSBCTSSCTSKUTS2R
SCHEMBL3902634 0.77 CTSS (0.49) CTSLCTSBCTSSCTSKMCL1
SCHEMBL3893070 0.76 CTSS (0.43) CTSLCTSBCTSSCTSKUTS2R
SCHEMBL3898975 0.75 CTSS (0.53) CTSLCTSBCTSSPPARGPPARA
SCHEMBL3893067 0.74 CTSK (0.43) CTSLCTSBCTSSCTSKUTS2R
SCHEMBL6567349 0.73 CTSS (0.47) CTSLCTSBCTSSCTSKUTS2R
SCHEMBL3910486 0.73 CTSL (0.46) CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO claimed
WO-2002100849-A2 NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-12-19 WO disclosed