SCHEMBL6567608

SCHEMBL6567608

CC(=O)C1CC(CC(=O)Nc2cc(Cl)c(O)c(Cl)c2)C1(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.39
P2RX5 Q93086 1/20 0.39
P2RX4 Q99571 1/20 0.39
P2RX2 Q9UBL9 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
DHODH Q02127 1/20 0.36
NPC1 O15118 2/20 0.35
GAA P10253 1/20 0.35
RAB9A P51151 1/20 0.35
LMNA P02545 4/20 0.34
MAP2K1 Q02750 1/20 0.34
CYP3A4 P08684 1/20 0.34
ABL1 P00519 2/20 0.34
RIN1 Q13671 2/20 0.34
TDP1 Q9NUW8 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6567255 0.70 EPHX2 (0.59) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL16150319 0.68 CYP3A4 (0.66) MEN1KMT2APOLBALDH1A1DHODH
SCHEMBL6567675 0.68 P2RX7 (0.65) P2RX7P2RX5P2RX4P2RX2MEN1
SCHEMBL6568487 0.68 ALDH1A1 (0.38) P2RX7P2RX5P2RX4P2RX2MEN1
SCHEMBL6566838 0.67 P2RX7 (0.53) P2RX7P2RX5P2RX4P2RX2MEN1
SCHEMBL16152426 0.66 GRM2 (0.38) GRM1
SCHEMBL4905385 0.66 GRM2 (0.38) GRM1
SCHEMBL4905394 0.66 GRM2 (0.38) GRM1
SCHEMBL18723739 0.66 GRM2 (0.38) GRM1
SCHEMBL6560389 0.66 GRM2 (0.38) GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed