SCHEMBL6570731

SCHEMBL6570731

COCCN(CCOC)c1ccc(N)c(-c2ccc(C(C)=O)cc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 1/20 0.38
F2 P00734 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
RELA Q04206 6/20 0.36
CHEK2 O96017 2/20 0.36
HSD17B1 P14061 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
OPRK1 P41145 1/20 0.35
UTS2R Q9UKP6 1/20 0.35
HDAC4 P56524 1/20 0.35
CREBBP Q92793 1/20 0.35
MMP12 P39900 1/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572668 0.90 RARB (0.43) F2PRSS1PRSS2PRSS3RELA
SCHEMBL6572986 0.87 HSD17B1 (0.39) HDAC2RELAHSD17B1CREBBPMEN1
SCHEMBL6571056 0.84 MGAM (0.36) F2PRSS1PRSS2PRSS3RELA
SCHEMBL6571429 0.84 ALDH1A1 (0.36) F2PRSS1PRSS2PRSS3RELA
SCHEMBL6571926 0.83 F2 (0.38) F2PRSS1PRSS2PRSS3MEN1
SCHEMBL6572008 0.83 MAPT (0.35) F2PRSS1PRSS2PRSS3CYP3A4
SCHEMBL6570799 0.83 GRM2 (0.38) HDAC2F2PRSS1PRSS2PRSS3
SCHEMBL6570859 0.83 S100B (0.37) F2PRSS1PRSS2PRSS3CYP3A4
SCHEMBL6571984 0.82 S100B (0.36) F2PRSS1PRSS2PRSS3CYP3A4
SCHEMBL6572323 0.82 ALOX15 (0.40) HDAC2RELACYP3A4CYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed