SCHEMBL6571392

SCHEMBL6571392

CNc1ccc(N)c(-c2ccccc2O)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.39
SMARCA2 P51531 2/20 0.38
SMARCA4 P51532 2/20 0.38
BRD4 O60885 1/20 0.38
NR1I2 O75469 1/20 0.38
PBRM1 Q86U86 1/20 0.38
TSHR P16473 2/20 0.38
ALOX15 P16050 2/20 0.38
HSD17B10 Q99714 2/20 0.37
IDO1 P14902 2/20 0.37
HDAC3 O15379 1/20 0.37
EP300 Q09472 1/20 0.37
KAT2B Q92831 1/20 0.37
KAT8 Q9H7Z6 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
ALDH1A1 P00352 5/20 0.36
GFER P55789 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572173 0.89 TP53 (0.41) TSHRALOX15HSD17B10EP300HSP90AA1
SCHEMBL3790053 0.85 ALDH1A1 (0.52) PDK2TSHRALOX15HSD17B10IDO1
SCHEMBL6571922 0.83 TSHR (0.41) PDK2TSHRALOX15HSD17B10ALDH1A1
SCHEMBL6572709 0.83 ALDH1A1 (0.41) ALOX15HSD17B10HSP90AA1HSP90AB1ALDH1A1
SCHEMBL6570909 0.81 PDE10A (0.44) TSHRALOX15HSD17B10IDO1HDAC3
SCHEMBL16961438 0.81 MAPT (0.50) ALOX15HSD17B10SMN1; SMN2ALDH1A1GFER
SCHEMBL6573100 0.81 NUDT1 (0.42) PDK2TSHRALOX15HSD17B10ALDH1A1
SCHEMBL6571996 0.80 ALDH1A1 (0.44) ALOX15HSD17B10HSP90AA1HSP90AB1ALDH1A1
SCHEMBL6572432 0.78 BRD4 (0.38) SMARCA2SMARCA4BRD4NR1I2PBRM1
SCHEMBL6571563 0.77 HTR7 (0.45) HSD17B10IDO1SMN1; SMN2HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed