SCHEMBL6571563

SCHEMBL6571563

CNc1ccc(N)c(-c2ccccc2OC)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 6/20 0.45
HSP90AA1 P07900 2/20 0.44
ALDH1A1 P00352 7/20 0.44
TDP1 Q9NUW8 2/20 0.44
ADRA2B P18089 1/20 0.44
PTGS1 P23219 1/20 0.44
HSD17B10 Q99714 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
MAPT P10636 2/20 0.41
MAPK1 P28482 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HTR1A P08908 2/20 0.41
HTR1D P28221 2/20 0.41
HTR1B P28222 2/20 0.41
HTR2A P28223 2/20 0.41
HTR1E P28566 2/20 0.41
HTR2B P41595 2/20 0.41
HTR5A P47898 2/20 0.41
HTR6 P50406 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572173 0.92 TP53 (0.41) HTR7HSP90AA1ALDH1A1TDP1ADRA2B
SCHEMBL6573517 0.84 NR3C1 (0.41) HTR7HSP90AA1ALDH1A1TDP1ADRA2B
SCHEMBL3790053 0.83 ALDH1A1 (0.52) ALDH1A1TDP1HSD17B10CYP3A4MAPT
SCHEMBL6571911 0.81 ALDH1A1 (0.49) HSP90AA1ALDH1A1HSD17B10CYP3A4MAPT
SCHEMBL6573246 0.80 GAA (0.43) HTR7ALDH1A1TDP1ADRA2BPTGS1
SCHEMBL6570699 0.80 ALDH1A1 (0.50) HTR7ALDH1A1TDP1ADRA2BPTGS1
SCHEMBL6570989 0.80 ALDH1A1 (0.50) HTR7HSP90AA1ALDH1A1TDP1ADRA2B
SCHEMBL6572475 0.78 HDAC4 (0.39) ALDH1A1TDP1HSD17B10CYP3A4MAPT
Hydrochloric Acid SCHEMBL6574711 0.78 ALDH1A1 (0.48) HTR7HSP90AA1ALDH1A1TDP1ADRA2B
SCHEMBL6573100 0.78 NUDT1 (0.42) ALDH1A1TDP1HSD17B10CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed