SCHEMBL6572572

SCHEMBL6572572

COCCN(CCOC)c1ccc(N)c(-c2ccc(O)cc2O)c1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 3/20 0.34
PDK1 Q15118 3/20 0.34
HSP90AA1 P07900 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
S100B P04271 1/20 0.33
PTPN1 P18031 1/20 0.31
TYR P14679 1/20 0.31
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
F2 P00734 1/20 0.30
PRSS1 P07477 1/20 0.30
PRSS2 P07478 1/20 0.30
PRSS3 P35030 1/20 0.30
SNCA P37840 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6572226 0.89 TSHR (0.37) S100BALDH1A1CYP3A4GAAF2
SCHEMBL6571124 0.86 F2 (0.36) S100BALDH1A1GAAF2PRSS1
SCHEMBL6571056 0.85 MGAM (0.36) S100BGAAF2PRSS1PRSS2
SCHEMBL6572717 0.83 ALOX5 (0.36) PDK1S100BTYRALDH1A1GAA
SCHEMBL6572336 0.82 S100B (0.33) S100BCYP3A4F2PRSS1PRSS2
SCHEMBL6571441 0.82 CYP3A4 (0.38) ALDH1A1CYP3A4F2PRSS1PRSS2
SCHEMBL6570734 0.81 S100B (0.34) S100BALDH1A1CYP3A4GAA
SCHEMBL6572395 0.77 CRHR1 (0.48) CYP3A4
SCHEMBL6572502 0.77 S100B (0.40) S100BALDH1A1GAAF2PRSS1
SCHEMBL6573203 0.77 ALDH1A1 (0.34) S100BALDH1A1GAAF2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP claimed
EP-1051143-B1 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AG (DE) 2004-07-21 EP disclosed
US-6500213-B1 Oxidizing hair coloring agents containing 2,5-diamino-1-phenylbenzene derivatives and novel 2,5-diamino-1-phenylbenzene derivatives WELLA AKTIENGESELLSCHAFT (DE) 2002-12-31 US disclosed
EP-1051143-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES Wella Aktiengesellschaft (DE) 2000-11-15 EP disclosed
WO-1999059527-A2 OXIDIZING HAIR COLORING AGENTS CONTAINING 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES AND NOVEL 2,5-DIAMINO-1-PHENYLBENZENE DERIVATIVES WELLA AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed