SCHEMBL657352

SCHEMBL657352

CC(=O)OCOC(=O)C(COC(C)=O)(C(=O)O)C(CC(=O)c1ccc(C(F)(F)F)cc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.47
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
LDHA P00338 1/20 0.37
LDHB P07195 1/20 0.37
HSD11B1 P28845 1/20 0.37
SLC6A9 P48067 2/20 0.35
PTPN1 P18031 2/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
GSK3B P49841 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 2/20 0.34
TSHR P16473 2/20 0.34
CYP2C19 P33261 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CACNA1A O00555 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL658836 0.91 UTS2R (0.39) PDPK1ALDH1A1MAPTLDHALDHB
SCHEMBL658601 0.88 PDPK1 (0.41) PDPK1MAPTCYP2C9CYP2C19MEN1
SCHEMBL657804 0.88 SRD5A2 (0.38) ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL659012 0.84 GLA (0.41) PDPK1ALDH1A1MAPTPTPN1CYP1A2
SCHEMBL656363 0.82 ALDH1A1 (0.45) ALDH1A1CYP1A2TSHRCYP2C19
SCHEMBL656175 0.79 KMT2A (0.47) PDPK1ALDH1A1MAPTCYP2C9CYP2C19
SCHEMBL657877 0.78 CYP2C9 (0.50) PDPK1ALDH1A1MAPTCYP2C9CYP2C19
SCHEMBL657976 0.78 PDPK1 (0.49) PDPK1CYP2C9KMT2ASMN1; SMN2
SCHEMBL657351 0.78 PDPK1 (0.67) PDPK1ALDH1A1MAPTLDHALDHB
SCHEMBL7109215 0.70 NPC1 (0.52) ALDH1A1MAPTTSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120046307-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2012-02-23 US claimed
US-8912186-B2 Allosteric protein kinase modulators UNIVERSITAET DES SAARLANDES (DE) 2014-12-16 US disclosed
US-20120046307-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2012-02-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046307-A1 ALLOSTERIC PROTEIN KINASE MODULATORS AURKC, AURKA, AURKB PDPK1 109/4885ALDH1A1 4784/4885MAPT 964/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.