SCHEMBL657437

SCHEMBL657437

O=C(Cl)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.52
ERCC1 P07992 4/20 0.50
ERCC4 Q92889 4/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
MAPK1 P28482 1/20 0.50
CYP2C19 P33261 1/20 0.50
P2RX7 Q99572 1/20 0.50
GALR3 O60755 1/20 0.49
NR2F2 P24468 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
GGPS1 O95749 1/20 0.49
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30321024 1.00 IDO1 (0.52) IDO1ERCC1ERCC4CYP1A2CYP3A4
SCHEMBL260323 0.86 L3MBTL1 (0.55) IDO1ERCC1ERCC4P2RX7TDP1
SCHEMBL29718886 0.86 L3MBTL1 (0.55) IDO1ERCC1ERCC4P2RX7TDP1
SCHEMBL28940593 0.85 IDO1 (0.54) IDO1ERCC1ERCC4CYP1A2CYP3A4
SCHEMBL29419329 0.83 CHRM1 (0.57) IDO1ERCC1ERCC4CYP1A2CYP3A4
SCHEMBL260512 0.83 CHRM1 (0.57) IDO1ERCC1ERCC4CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL2532568 0.82 CHRM1 (0.55) IDO1ERCC1ERCC4CYP2C9P2RX7
SCHEMBL20796876 0.82 GALR3 (0.55) IDO1ERCC1ERCC4CYP1A2CYP3A4
SCHEMBL29712851 0.82 IDO1 (0.50) IDO1ERCC1ERCC4CYP1A2CYP3A4
SCHEMBL4686080 0.82 IDO1 (0.50) IDO1ERCC1ERCC4CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 139 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109369587-A A kind of production technology of high-purity high-yield Envidor 新沂市永诚化工有限公司 2019-02-22 CN claimed
CN-109053410-A It is a kind of synthesize 1- hydroxy-cyclohexyl formic acid new process and application 兰博尔开封科技有限公司 2018-12-21 CN claimed
CN-108863774-A A kind of 2,4 dichloro benzene chloroacetic chloride synthetic method 石家庄市绿丰化工有限公司 2018-11-23 CN claimed
CN-108658913-A A kind of method of synthetic pesticide Envidor key intermediate 石家庄市绿丰化工有限公司 2018-10-16 CN claimed
US-20240417379-A1 P2X4 RECEPTOR ANTAGONIST NIPPON CHEMIPHAR CO., LTD (JP) 2024-12-19 US disclosed
US-12116351-B2 P2X4 receptor antagonist NIPPON CHEMIPHAR CO., LTD (JP) 2024-10-15 US disclosed
CN-113880764-B Sinomenine derivative and preparation method and application thereof 北京师范大学 2023-04-18 CN disclosed
US-11584744-B2 Inhibitors of type 1 methionyl-tRNA synthetase and methods of using them UNIVERSITY OF WASHINGTON (US) 2023-02-21 US disclosed
US-11584744-B2 Inhibitors of type 1 methionyl-tRNA synthetase and methods of using them UNIVERSITY OF WASHINGTON (US) 2023-02-21 US disclosed
US-20220380322-A1 P2X4 RECEPTOR ANTAGONIST NIPPON CHEMIPHAR CO., LTD (JP) 2022-12-01 US disclosed
US-11434207-B2 P2X4 receptor antagonist NIPPON CHEMIPHAR CO., LTD (JP) 2022-09-06 US disclosed
CN-113880764-A Sinomenine derivative and preparation method and application thereof 北京师范大学 2022-01-04 CN disclosed
US-4262072-A ABRASION RESISTANT MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1981-04-14 US disclosed
US-4258189-A ANTHRAPYRIDINE MODIFIED ADDITION POLYMERS DYNAPOL (US) 1981-03-24 US disclosed
US-4249011-A CURING AGENTS FOR ADDITION PHOTOPOLYMERIZATION MINNESOTA MINING AND MANUFACTURING COMPANY 1981-02-03 US disclosed
WO-1981000011-A1 POLY(ETHYLENICALLY UNSATURATED ALKOXY)HETEROCYCLIC COMPOUNDS AND CROSSLINKED POLYMERIC COATINGS MINNESOTA MINING & MFG (US) 1981-01-08 WO disclosed
EP-0006254-A1 Benzoin oxime derivatives, process for their preparation, compositions containing such derivatives and method for their use as fungicides SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1980-01-09 EP disclosed
US-4073936-A Hypolipidemic allene carboxylic esters SANDOZ, INC. (US) 1978-02-14 US disclosed
US-4011339-A ANTIINFLAMMATORY AGENTS SANDOZ, INC. (US) 1977-03-08 US disclosed
US-3992396-A TRANQUILIZERS, HYPNOTICS SANDOZ, INC. (US) 1976-11-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220380322-A1 P2X4 RECEPTOR ANTAGONIST P2RX7, P2RX1, P2RX2 IDO1 1912/4885ERCC1 4026/4885ERCC4 4269/4885
US-20240417379-A1 P2X4 RECEPTOR ANTAGONIST P2RX7, P2RX1, P2RX2 IDO1 1876/4885ERCC1 3024/4885ERCC4 3623/4885
US-12116351-B2 P2X4 receptor antagonist P2RX7, P2RX1, P2RX2 IDO1 1912/4885ERCC1 4026/4885ERCC4 4269/4885
US-11434207-B2 P2X4 receptor antagonist P2RX7, P2RX1, P2RX2 IDO1 1912/4885ERCC1 4026/4885ERCC4 4269/4885
US-11584744-B2 Inhibitors of type 1 methionyl-tRNA synthetase and methods of using them AARS1, EMG1, GARS1 IDO1 1989/4885ERCC1 3093/4885ERCC4 2208/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.