SCHEMBL6578559

SCHEMBL6578559

COc1ccc(-c2nc(-c3cccc(C=O)c3)n(C3CCCC3)n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNJ6 P48051 2/20 0.41
KCNJ5 P48544 2/20 0.41
KCNJ3 P48549 2/20 0.41
AVPR1B P47901 10/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
LMNA P02545 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6580712 0.96 NR1H2 (0.40) KCNJ6KCNJ5KCNJ3AVPR1BPDE4A
SCHEMBL6581016 0.84 AVPR1B (0.43) AVPR1B
SCHEMBL6582832 0.82 L3MBTL1 (0.43) AVPR1B
SCHEMBL6580839 0.81 KDM4C (0.49) NPC1RAB9ATDP1ALDH1A1HPGD
SCHEMBL6580805 0.81 TGM2 (0.51) AVPR1BNPC1RAB9ATDP1ALDH1A1
SCHEMBL6581299 0.80 NR1H2 (0.45) AVPR1BNPC1RAB9ATDP1ALDH1A1
SCHEMBL6582750 0.80 NR1H2 (0.46) AVPR1BNPC1RAB9ATDP1ALDH1A1
Hydrochloric Acid SCHEMBL6583804 0.79 HTR7 (0.41) KCNJ6KCNJ5KCNJ3AVPR1BPDE4A
SCHEMBL6581102 0.79 NR1H3 (0.57) AVPR1BNPC1RAB9ATDP1ALDH1A1
SCHEMBL6582793 0.78 NR1H2 (0.47) AVPR1BNPC1RAB9ATDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed