SCHEMBL6580414

SCHEMBL6580414

NOC(=O)C(CCCc1ccccc1)CS(=O)(=O)C1CCN(C(=O)c2ccccc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.44
CA12 O43570 2/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
CA7 P43166 1/20 0.42
CA14 Q9ULX7 1/20 0.42
KMT2A Q03164 4/20 0.41
KCNH2 Q12809 2/20 0.41
MEN1 O00255 2/20 0.41
CAPN1 P07384 1/20 0.41
HTR2A P28223 1/20 0.41
MMP1 P03956 2/20 0.41
MMP2 P08253 2/20 0.41
MMP3 P08254 2/20 0.41
MMP9 P14780 2/20 0.41
MMP8 P22894 2/20 0.41
ADRB3 P13945 1/20 0.40
EPHX1 P07099 1/20 0.40
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydroxyamine SCHEMBL6580410 0.89 MMP1 (0.50) SIGMAR1CA12CA1CA2CA9
SCHEMBL6581071 0.89 MMP1 (0.52) SIGMAR1CA12CA1CA2CA9
SCHEMBL6575904 0.85 MMP1 (0.55) SIGMAR1CA12CA1CA2CA9
SCHEMBL6578067 0.75 STS (0.52) MMP1MMP2MMP3MMP9MMP8
SCHEMBL6580383 0.74 HTR2A (0.50) SIGMAR1KMT2AKCNH2MEN1HTR2A
SCHEMBL7079165 0.73 MMP2 (0.54) MMP1MMP2MMP3MMP9MMP8
SCHEMBL6578667 0.72 STS (0.51) MMP1MMP2MMP3MMP9MMP8
SCHEMBL6578105 0.71 SIGMAR1 (0.49) SIGMAR1KMT2AKCNH2MEN1MMP1
SCHEMBL6578655 0.71 MMP2 (0.53) SIGMAR1KCNH2HTR2AMMP1MMP2
SCHEMBL27740557 0.70 GRIK1 (0.55) MMP1MMP2MMP3MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968182-B1 HYDROXAMIC AND CARBOXYLIC ACID DERIVATIVES HAVING MMP AND TNF INHIBITORY ACTIVITY DARWIN DISCOVERY LTD (GB) 2004-05-06 EP claimed