SCHEMBL6581048

SCHEMBL6581048

COc1ccc(-c2nc(-c3cccc(CN(C)C)c3)n(C)n2)cc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 1/20 0.46
CSF1R P07333 1/20 0.45
AVPR1B P47901 1/20 0.45
S1PR1 P21453 1/20 0.43
HSD17B2 P37059 1/20 0.42
PSEN1 P49768 2/20 0.42
PSEN2 P49810 2/20 0.42
APH1B Q8WW43 2/20 0.42
NCSTN Q92542 2/20 0.42
APH1A Q96BI3 2/20 0.42
PSENEN Q9NZ42 2/20 0.42
TDP2 O95551 1/20 0.40
TLR8 Q9NR97 2/20 0.40
TLR7 Q9NYK1 2/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
TLR9 Q9NR96 1/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584053 0.84 ACP1 (0.46) HTR7AVPR1BHSD17B2ADORA2AADORA1
Hydrochloric Acid SCHEMBL6580533 0.83 ACP1 (0.45) HTR7AVPR1BHSD17B2ADORA2AADORA1
SCHEMBL6581290 0.81 NR1H2 (0.50) HTR7S1PR1HSD17B2TDP2ADORA2A
Hydrochloric Acid SCHEMBL6580743 0.80 NR1H2 (0.49) HTR7S1PR1HSD17B2TDP2ADORA2A
SCHEMBL6580847 0.79 TDP2 (0.44) HSD17B2PSEN1PSEN2APH1BNCSTN
SCHEMBL6580791 0.78 TNK2 (0.43) HTR7AVPR1BS1PR1HSD17B2ADORA2A
SCHEMBL6580942 0.78 HTR7 (0.46) HTR7CSF1RS1PR1PSEN1PSEN2
Hydrochloric Acid SCHEMBL6581027 0.77 HTR7 (0.46) HTR7CSF1RS1PR1PSEN1PSEN2
Hydrochloric Acid SCHEMBL6583998 0.77 TNK2 (0.42) HTR7AVPR1BS1PR1HSD17B2ADORA2A
Hydrochloric Acid SCHEMBL6580650 0.72 NR1H3 (0.52) HTR7AVPR1BS1PR1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP claimed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US claimed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP claimed
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed