SCHEMBL6581263

SCHEMBL6581263

CC(C)(C)OC(=O)c1cccc(NCC(=O)N2CCC(CNCc3ccncc3)CC2)c1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SCD O00767 12/20 0.45
TGFBR1 P36897 1/20 0.37
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRM5 P41594 1/20 0.36
SLC2A1 P11166 1/20 0.36
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6582688 0.90 CYP2D6 (0.44) SCDTGFBR1ADRA1AADRA1BCYP2D6
SCHEMBL6582672 0.76 GRIN2B (0.39) SCDADRA1AADRA1BCYP2D6CYP2C9
SCHEMBL6581653 0.75 HTR1A (0.37)
Hydrochloric Acid SCHEMBL6582680 0.75 F10 (0.45) SCDCYP2D6CYP2C9GRIN2BSLC2A1
SCHEMBL6584670 0.74 HTR1A (0.37)
SCHEMBL5867949 0.73 MEN1 (0.38) ADRA1AADRA1BCYP2D6KDM4EPKM
SCHEMBL6583196 0.71 BRD4 (0.38) SCDTGFBR1ADRA1AADRA1BGRIN2B
Hydrochloric Acid SCHEMBL6582721 0.71 F10 (0.40) SCDCYP2C9GRIN2BSLC2A1KDM4E
SCHEMBL6582799 0.71 CCNT1 (0.38) SCDTGFBR1CYP2D6CYP2C9GRIN2B
SCHEMBL6582859 0.70 GRIN2B (0.46) SCDCYP2D6CYP2C9GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1455788-A1 1-GLYCINYL-4-AMINOMETHYL-PIPERIDINE DERIVATIVES AS FACTOR XA INHIBITORS ELI LILLY AND COMPANY (US) 2004-09-15 EP disclosed
WO-2003049737-A1 CHEMICAL COMPOUNDS ELI LILLY AND COMPANY (US) 2003-06-19 WO disclosed