SCHEMBL6581350

SCHEMBL6581350

CNCC(=O)Nc1ccc(Cl)c(COc2ccc3nc(C)ccc3c2)c1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 2/20 0.37
KLKB1 P03952 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
KCNH2 Q12809 3/20 0.35
TP53 P04637 1/20 0.35
KDM4E B2RXH2 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
LMNA P02545 1/20 0.34
BLM P54132 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7906001 0.80 BDKRB2 (0.54) BDKRB2MAPTALDH1A1HPGDLMNA
SCHEMBL6578780 0.77 NCF1 (0.40) KLKB1KDM4ENPC1RAB9AMAPT
SCHEMBL6576127 0.75 S1PR4 (0.42) KLKB1TP53NPC1RAB9AKMT2A
SCHEMBL6936592 0.69 KDM4E (0.42) KDM4ENPC1RAB9AMAPTALDH1A1
SCHEMBL8097174 0.69 BDKRB2 (0.40) BDKRB2KLKB1KDM4ERAB9AALDH1A1
SCHEMBL6581385 0.68 TP53 (0.42) TP53NPC1MEN1KMT2AMAPT
SCHEMBL6935565 0.67 BDKRB2 (0.46) BDKRB2
SCHEMBL6580627 0.66 NCF1 (0.41) KDM4EMAPTALDH1A1GAATSHR
SCHEMBL6576073 0.66 KDM4E (0.38) KDM4ENPC1RAB9AMEN1KMT2A
SCHEMBL8098950 0.66 S1PR4 (0.37) BDKRB2KLKB1KDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0867432-B1 Fused N-heterocyclic compounds substituted with benzyloxy, process for their preparation and their use as bradykinin receptor antagonists AVENTIS PHARMA GMBH (DE) 2004-06-09 EP disclosed
EP-0867432-A2 Fused N-heterocyclic compounds substituted with benzyloxy, process for their preparation and their use as bradykinin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-09-30 EP disclosed