SCHEMBL6581393

SCHEMBL6581393

O=C(O)n1c(=O)ccc2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.52
BRD4 O60885 1/20 0.52
BRPF1 P55201 1/20 0.52
CA9 Q16790 1/20 0.52
KAT2B Q92831 1/20 0.52
BRD9 Q9H8M2 1/20 0.52
TSHR P16473 2/20 0.42
KMT2A Q03164 2/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NOTUM Q6P988 1/20 0.40
DAO P14920 1/20 0.39
MCL1 Q07820 1/20 0.38
P2RX4 Q99571 1/20 0.38
APEX1 P27695 1/20 0.37
ALDH1A1 P00352 2/20 0.37
POLB P06746 1/20 0.35
LMNA P02545 1/20 0.35
IDO1 P14902 1/20 0.35
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10662835 0.86 CA12 (0.53) CA12BRD4BRPF1CA9KAT2B
SCHEMBL6195893 0.85 RAB9A (0.56) CA12BRD4BRPF1CA9KAT2B
SCHEMBL30804587 0.85 RAB9A (0.56) CA12BRD4BRPF1CA9KAT2B
SCHEMBL30672091 0.82 CA12 (0.55) CA12BRD4BRPF1CA9KAT2B
SCHEMBL6568800 0.82 CA12 (0.55) CA12BRD4BRPF1CA9KAT2B
SCHEMBL28320396 0.79 KCNMA1 (0.44) CA12BRD4BRPF1CA9KAT2B
SCHEMBL30321500 0.78 CA12 (0.50) CA12BRD4BRPF1CA9KAT2B
SCHEMBL27637776 0.78 CA12 (0.42) CA12BRD4BRPF1CA9KAT2B
SCHEMBL27916356 0.78 CA12 (0.42) CA12BRD4BRPF1CA9KAT2B
SCHEMBL27485103 0.76 KMO (0.41) MCL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 207 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107056810-B A kind of preparation method of Carbostyril carboxylic acid derivatives 广东省中医院 2019-04-26 CN claimed
CN-107056810-A A kind of preparation method of Carbostyril carboxylic acid derivatives 广东省中医院 2017-08-18 CN claimed
CN-106687179-A Methods for treating infections 梅琳塔治疗公司 2017-05-17 CN claimed
CN-106572982-A Antimicrobial compositions with effervescent agents 梅琳塔治疗公司 2017-04-19 CN claimed
CN-106237335-A A kind of dermatological field antibacterial 陈广圣 2016-12-21 CN claimed
CN-102215690-A Antimicrobial compositions RIB X PHARMACEUTICALS INC 2011-10-12 CN claimed
CN-101817820-B Method for synthesizing moxifloxacin hydrochloride CHONGQING BOTENG FINE CHEMICAL CO LTD 2011-10-05 CN claimed
CN-101817820-A Method for synthesizing moxifloxacin hydrochloride CHONGQING BOTENG FINE CHEMICAL CO LTD 2010-09-01 CN claimed
CN-100410249-C 7-(4-substituted 3- cyclopropylaminomethyl-1- pyrrolidinyl) Q uinolonecarboxylic acid derivative KYORIN SEIYAKU KK (JP) 2008-08-13 CN claimed
CN-100395244-C Quinolone carboxylic acid derivatives or their salts TOYAMA CHEMICAL CO LTD (JP) 2008-06-18 CN claimed
CN-1035945-C 5-Alkylquinolonecarboxylic acids BAYER AG (DE) 1997-09-24 CN claimed
CN-1128995-A Novel Quinolone carboxylic acid derivative DONG WHA PHARM IND CO LTD (KR) 1996-08-14 CN claimed
CN-1111629-A 5-vinyl-, 5-ethynylquinolone-and 5-vinyl-, 5-ethynylnaphthyridonecarboxylic acids BAYER AG (DE) 1995-11-15 CN claimed
CN-1108968-A Use of ion exchange resins loaded with quioolonecarboxylic acid derivatives BAYER AG (DE) 1995-09-27 CN claimed
CN-1094405-A New Carbostyril carboxylic acid derivatives and preparation method thereof KOREA RES INST CHEM TECH (KR) 1994-11-02 CN claimed
CN-1046162-A The 5-Alkylquinolonecarboxacids acids BAYER AG (DE) 1990-10-17 CN claimed
CN-1037335-A The preparation method of 1-cyclopropyl Quinolone carboxylic acid and derivative thereof BAYER AG (DE) 1989-11-22 CN claimed
CN-1037147-A N-cyclopropyl aniline and the application in preparation 1-cyclopropyl quinolone carboxylic acid and its derivative thereof BAYER AG (DE) 1989-11-15 CN claimed
CN-88103473-A Preparation and application of ion exchange resin loaded with quinolone carboxylic acid derivative 1988-12-28 CN claimed
CN-86104256-A 1, the preparation method of 8-bridging 4-quinolone-3-carboxylic-acid 1987-03-18 CN claimed