SCHEMBL6581698

SCHEMBL6581698

CCCC1(c2ccccc2)CC(Nc2n[nH]cc2OC(=O)OCC)C(=O)O1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.32
TYMS P04818 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
HTT P42858 2/20 0.32
OPRM1 P35372 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31
ELANE P08246 2/20 0.30
MAPT P10636 2/20 0.30
TSHR P16473 2/20 0.30
ALOX5 P09917 1/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MEN1 O00255 2/20 0.30
CYP1A2 P05177 2/20 0.30
CYP2C19 P33261 2/20 0.30
KMT2A Q03164 2/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6579675 0.95 TYMS (0.32) ALDH1A1TYMSSMN1; SMN2L3MBTL1HTT
SCHEMBL6291868 0.86 KMT2A (0.36) ALDH1A1SMN1; SMN2HTTPOLBRAB9A
SCHEMBL6291852 0.81 CNR2 (0.35) ALDH1A1SMN1; SMN2L3MBTL1HTTRAB9A
SCHEMBL6585426 0.81 HPGDS (0.33) ALDH1A1SMN1; SMN2RAB9AMAPTALOX5
SCHEMBL6152031 0.77 OPRM1 (0.32) OPRM1
SCHEMBL5776518 0.74 OPRM1 (0.31) ALDH1A1L3MBTL1OPRM1MAPTLMNA
SCHEMBL6581680 0.72 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2L3MBTL1HTTPOLB
SCHEMBL6288865 0.71 TSHR (0.31) TSHRNPSR1KMT2A
SCHEMBL5773302 0.70 MAPK1 (0.30)
SCHEMBL5775977 0.70 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2L3MBTL1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406888-A1 SUBSTITUTED $G(G)-LACTONE COMPOUNDS SERVING AS NMDA ANTAGONISTS Grünenthal GmbH (DE) 2004-04-14 EP claimed
WO-2003004483-A1 SUBSTITUTED $G(G)-LACTONE COMPOUNDS SERVING AS NMDA ANTAGONISTS Grünenthal GmbH (DE) 2003-01-16 WO claimed
EP-1406888-A1 SUBSTITUTED $G(G)-LACTONE COMPOUNDS SERVING AS NMDA ANTAGONISTS Grünenthal GmbH (DE) 2004-04-14 EP disclosed
WO-2003004483-A1 SUBSTITUTED $G(G)-LACTONE COMPOUNDS SERVING AS NMDA ANTAGONISTS Grünenthal GmbH (DE) 2003-01-16 WO disclosed