SCHEMBL6583477

SCHEMBL6583477

COc1ccc(C2=CC(N)(C(=O)C(C)c3ccc(CC(C)C)cc3)N=N2)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.45
CXCR1 P25024 3/20 0.41
CXCR2 P25025 3/20 0.41
TPH1 P17752 2/20 0.39
FAAH O00519 3/20 0.38
PTGS1 P23219 4/20 0.38
PTGS2 P35354 3/20 0.38
LMNA P02545 2/20 0.38
CYP2C9 P11712 2/20 0.38
AKR1C3 P42330 2/20 0.38
ALB P02768 1/20 0.38
ESR1 P03372 1/20 0.38
ALOX5 P09917 1/20 0.38
RARB P10826 1/20 0.38
ADRB3 P13945 1/20 0.38
NFKB1 P19838 1/20 0.38
HTR2A P28223 1/20 0.38
NR1I3 Q14994 1/20 0.38
SLC22A6 Q4U2R8 1/20 0.38
CXCL8 P10145 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584448 0.71 NPY5R (0.52) LMNACYP2C9
SCHEMBL6584786 0.71 PTGS2 (0.43) PTGS1PTGS2LMNACYP2C9AKR1C3
SCHEMBL6583482 0.69 EPHX1 (0.43) EPHX1CXCR1CXCR2TPH1FAAH
SCHEMBL6585213 0.69 NPY5R (0.55) CXCR1CXCR2FAAHLMNACHRM1
SCHEMBL3152241 0.66 EPHX1 (1.00) EPHX1CXCR1CXCR2FAAHPTGS1
SCHEMBL260688 0.66 EPHX1 (1.00) EPHX1CXCR1CXCR2FAAHPTGS1
SCHEMBL1883571 0.66 EPHX1 (1.00) EPHX1CXCR1CXCR2FAAHPTGS1
Hydrochloric Acid SCHEMBL3424822 0.65 EPHX1 (0.96) EPHX1CXCR1CXCR2FAAHPTGS1
SCHEMBL11570387 0.63 PTGS2 (0.56) EPHX1CXCR1CXCR2FAAHPTGS1
SCHEMBL5080304 0.63 PTGS2 (0.56) EPHX1CXCR1CXCR2FAAHPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945440-B1 AMINOPYRAZOLE DERIVATIVES BANYU PHARMA CO LTD (JP) 2004-05-26 EP claimed