SCHEMBL6584133

SCHEMBL6584133

COc1ccc(CCC2OC(=O)NC2=O)cc1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
NFKB1 P19838 1/20 0.49
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
APEX1 P27695 1/20 0.48
KMT2A Q03164 1/20 0.48
TUBB4A P04350 3/20 0.47
TUBB P07437 3/20 0.47
TUBA3C P0DPH7 3/20 0.47
TUBA1B P68363 3/20 0.47
TUBA4A P68366 3/20 0.47
TUBB4B P68371 3/20 0.47
TUBB3 Q13509 3/20 0.47
TUBB2A Q13885 3/20 0.47
TUBB8 Q3ZCM7 3/20 0.47
TUBA3E Q6PEY2 3/20 0.47
TUBA1A Q71U36 3/20 0.47
TUBA1C Q9BQE3 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8896521 0.92 TUBB4A (0.51) TSHRCYP1A2CYP3A4NFKB1MEN1
SCHEMBL6583808 0.90 TAAR1 (0.50) TSHRCYP1A2CYP3A4NFKB1LMNA
SCHEMBL8172780 0.87 GAA (0.47) TSHRCYP1A2CYP3A4NFKB1MEN1
SCHEMBL6583021 0.83 PPARG (0.51) TSHRCYP1A2CYP3A4NFKB1LMNA
SCHEMBL6584822 0.82 PPARG (0.49) TSHRCYP1A2CYP3A4NFKB1LMNA
SCHEMBL6583789 0.81 GAA (0.46) TSHRMEN1KMT2AGAAPPARG
SCHEMBL6583544 0.79 SIRT2 (0.59) CYP1A2CYP3A4MEN1LMNAKMT2A
SCHEMBL8175426 0.77 SHBG (0.52) TSHRCYP1A2CYP3A4NFKB1MEN1
SCHEMBL8890406 0.77 CA3 (0.42) LMNAKMT2AALDH1A1CA2
SCHEMBL6583749 0.76 PPARG (0.47) TSHRCYP3A4TUBB4ATUBBTUBA3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0710659-B1 Oxazolidinedione derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2004-01-28 EP disclosed
WO-1997000249-A1 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-03 WO disclosed
EP-0710659-A1 Oxazolidinedione derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-08 EP disclosed