SCHEMBL6585559

SCHEMBL6585559

COc1ccc(C2=CC(N)(C(=O)CCc3ccc4ccccc4c3)N=N2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CYP1A2 P05177 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
MAOA P21397 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HCAR2 Q8TDS4 1/20 0.39
BACE1 P56817 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
PKM P14618 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6585131 0.83 MTNR1A (0.46) MAPTMEN1KMT2ABACE1ALDH1A1
SCHEMBL6584448 0.79 NPY5R (0.52) LMNACYP1A2NPC1RAB9AKDM4E
SCHEMBL6588483 0.77 NPY5R (0.47) CYP1A2KDM4ESLC6A3MEN1KMT2A
SCHEMBL6583451 0.76 MC4R (0.37) NPC1RAB9AMAPTSLC6A3KMT2A
SCHEMBL6587116 0.76 NPC1 (0.37) LMNASMN1; SMN2CYP1A2NPC1RAB9A
SCHEMBL6584786 0.76 PTGS2 (0.43) LMNACYP1A2MAPTUTS2R
SCHEMBL6585427 0.75 NPY5R (0.42) LMNACYP1A2KDM4ECYP3A4MEN1
SCHEMBL6584761 0.73 RIOK2 (0.38) SLC6A3BACE1GSK3AMAPK10RIOK2
SCHEMBL28658857 0.71 NPC1 (0.70) LMNASMN1; SMN2CYP1A2NPC1RAB9A
SCHEMBL6588259 0.69 RIOK2 (0.38) SMN1; SMN2SLC6A3MEN1KMT2ARIOK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0945440-B1 AMINOPYRAZOLE DERIVATIVES BANYU PHARMA CO LTD (JP) 2004-05-26 EP claimed