SCHEMBL6586473

SCHEMBL6586473

CCOC(C)n1c(CN2CCCNCC2)nc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 4/20 0.49
ALDH1A1 P00352 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CXCR4 P61073 1/20 0.42
NR1I2 O75469 1/20 0.40
ABCB11 O95342 1/20 0.40
LMNA P02545 1/20 0.40
ESR1 P03372 1/20 0.40
PGR P06401 1/20 0.40
CYP3A4 P08684 1/20 0.40
PKM P14618 1/20 0.40
TSHR P16473 1/20 0.40
ADRA2B P18089 1/20 0.40
HTR2A P28223 1/20 0.40
ADRA1A P35348 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583159 0.96 HIF1A (0.46) HIF1AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL18306578 0.81 POLB (0.51) HIF1AALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL8315846 0.81 HTR3A (0.49)
SCHEMBL6583086 0.78 GRM2 (0.61) ALDH1A1LMNAMAPTNPSR1KDM4E
SCHEMBL8313269 0.78 HTR3A (0.53)
SCHEMBL6586477 0.77 MEN1 (0.54) ALDH1A1MEN1KMT2ALMNATSHR
SCHEMBL6962681 0.74 POLB (0.47) ALDH1A1MEN1KMT2ALMNATSHR
SCHEMBL6585574 0.72 GRM2 (0.67) ALDH1A1LMNAMAPTNPSR1KDM4E
SCHEMBL14602996 0.72 LMNA (0.61) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7481715 0.71 GRM2 (0.65) ALDH1A1LMNAMAPTNPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-B1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME KOWA CO (JP) 2004-10-27 EP disclosed
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed