SCHEMBL6586716

SCHEMBL6586716

NC1CCN(CC2CCN(C(=O)N3CCCCC3)CC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.54
CHRM5 P08912 1/20 0.44
ADRA2C P18825 1/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 9/20 0.43
TP53 P04637 1/20 0.43
THRB P10828 3/20 0.41
LMNA P02545 3/20 0.40
ACHE P22303 1/20 0.40
GAA P10253 1/20 0.39
HSD11B1 P28845 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584309 0.98 SMN1; SMN2 (0.51) SMN1; SMN2CHRM5ADRA2CALDH1A1MAPT
SCHEMBL14275787 0.84 ALDH1A1 (0.61) SMN1; SMN2ALDH1A1TP53LMNAHSD11B1
SCHEMBL382920 0.82 ALDH1A1 (0.56) ALDH1A1TP53HSD11B1
SCHEMBL6585178 0.81 SMN1; SMN2 (0.42) SMN1; SMN2CHRM5ADRA2CMAPTTP53
SCHEMBL6584534 0.80 CXCR3 (0.45) SMN1; SMN2MAPTTHRBLMNAACHE
SCHEMBL6586007 0.77 POLB (0.47) MAPTTP53THRBLMNAGAA
SCHEMBL6589869 0.77 CHRM5 (0.67) SMN1; SMN2CHRM5ADRA2CACHE
SCHEMBL1586529 0.77 CHRM5 (0.67) SMN1; SMN2CHRM5ADRA2CACHE
SCHEMBL11545422 0.77 CHRM5 (0.67) SMN1; SMN2CHRM5ADRA2CACHE
SCHEMBL1136825 0.76 GNAI3 (0.46) ALDH1A1TP53HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076055-B1 1- (1-SUBSTITUTED-4-PIPERIDINYL)METHYL]-4-PIPERIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, MEDICINAL COMPOSITIONS CONTAINING THE SAME AND INTERMEDIATES OF THESE COMPOUNDS DAINIPPON PHARMACEUTICAL CO (JP) 2004-11-24 EP disclosed
US-6294555-B1 SEROTONIN HT3 RECEPTOR ANTAGONIST FOR GASTROINTESTINAL DISORDERS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2001-09-25 US disclosed
EP-1076055-A1 1- (1-SUBSTITUTED-4-PIPERIDINYL)METHYL]-4-PIPERIDINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, MEDICINAL COMPOSITIONS CONTAINING THE SAME AND INTERMEDIATES OF THESE COMPOUNDS Dainippon Pharmaceutical Co., Ltd. (JP) 2001-02-14 EP disclosed