SCHEMBL6586759

SCHEMBL6586759

COC(=O)CS(=O)(=O)N1CCC(Cc2ccccc2)CC1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.60
MEN1 O00255 3/20 0.60
KMT2A Q03164 3/20 0.60
LMNA P02545 1/20 0.60
GAA P10253 1/20 0.60
HTT P42858 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.57
ALDH1A1 P00352 3/20 0.56
HPGD P15428 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
HSD17B10 Q99714 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
MMP2 P08253 1/20 0.54
MMP13 P45452 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6795444 0.85 MEN1 (0.61) MAPTMEN1KMT2ALMNASMN1; SMN2
SCHEMBL6585983 0.83 MMP3 (0.62) MAPTMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL14452167 0.82 MEN1 (0.61) MEN1KMT2ASMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL6588226 0.82 MMP3 (0.60) MAPTALDH1A1HPGDNPSR1HSD17B10
SCHEMBL14452185 0.79 MEN1 (0.58) MAPTMEN1KMT2ALMNASMN1; SMN2
SCHEMBL25094668 0.79 KDM4E (0.58) MEN1KMT2ALMNAALDH1A1L3MBTL1
SCHEMBL6584929 0.78 MMP3 (0.72) MAPTLMNAGAAALDH1A1HPGD
SCHEMBL7072831 0.77 MMP2 (0.73) MAPTMEN1KMT2ALMNAGAA
SCHEMBL14452149 0.77 MEN1 (0.58) MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL19201201 0.76 NCF1 (0.39) MAPTGAASMN1; SMN2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036062-B1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE (MMP) INHIBITORS PFIZER LTD (GB) 2004-01-02 EP disclosed
US-6495568-B1 TREATMENT OF TISSUE ULCERATION, WOUND REPAIR AND SKIN DISEASES WARNER-LAMBERT COMPANY 2002-12-17 US disclosed
CN-1362954-A Sulfamidohydroxamic acid metalloprotease inhibitor SEARLE & CO (US) 2002-08-07 CN disclosed
EP-1036062-A1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE (MMP) INHIBITORS Pfizer Limited (GB) 2000-09-20 EP disclosed
WO-1999029667-A1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE (MMP) INHIBITORS PFIZER LIMITED (GB) 1999-06-17 WO disclosed