SCHEMBL6587607

SCHEMBL6587607

Cc1c(O)ncnc1-c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIT P10721 9/20 0.41
ACACB O00763 1/20 0.37
MAPK14 Q16539 2/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CFTR P13569 1/20 0.36
KMO O15229 1/20 0.36
SLC34A1 Q06495 1/20 0.35
F9 P00740 1/20 0.35
F11 P03951 1/20 0.35
F7 P08709 1/20 0.35
CYP2C9 P11712 1/20 0.35
DHODH Q02127 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16281521 0.81 ADORA2A (0.46) KDM4EALDH1A1HTTSMN1; SMN2KMO
SCHEMBL6590702 0.74 EGLN1 (0.46) MAPK14KDM4EALDH1A1LMNACYP2C9
SCHEMBL2232292 0.70
SCHEMBL9748838 0.69 MAPK14 (0.46) MAPK14
SCHEMBL29811067 0.69 KMO (0.46) KITKMOF9
SCHEMBL16163570 0.68 KDR (0.51) KITKDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL12888433 0.67 RAB9A (0.44) MAPK14KDM4EALDH1A1LMNAHTT
SCHEMBL23147522 0.67 KMO (0.61) KITKMODHODH
SCHEMBL19933585 0.66 KMO (0.44) KITMAPK14KDM4ELMNASMN1; SMN2
SCHEMBL11713861 0.66 ACHE (0.46) KITMAPK14KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0781766-B1 HETEROCYCLIC DERIVATIVE AND MEDICINE NIPPON SHINYAKU CO LTD (JP) 2004-03-31 EP disclosed
US-6191149-B1 DRUG FOR CEREBROVASCULAR DISEASE NIPPON SHINYAKU, CO., LTD. (JP) 2001-02-20 US disclosed
US-5945426-A PREVENT NEURONAL DEATH NIPPON SHINYAKU CO., LTD. (JP) 1999-08-31 US disclosed
EP-0781766-A1 HETEROCYCLIC DERIVATIVE AND MEDICINE NIPPON SHINYAKU COMPANY, LIMITED (JP) 1997-07-02 EP disclosed