SCHEMBL6589528

SCHEMBL6589528

CCCC1(OC(=O)/C=C\C(=O)OC2(CCC)c3ccccc3CN2c2ccncc2)c2ccccc2CN1c1ccncc1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 2/20 0.32
MMP1 P03956 1/20 0.32
MMP3 P08254 1/20 0.32
ADAM17 P78536 1/20 0.32
ADAM9 Q13443 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
EED O75530 1/20 0.30
SLC6A2 P23975 1/20 0.30
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6592827 0.91 ALDH1A1 (0.33) MMP9MMP1MMP3ADAM17ADAM9
SCHEMBL8433460 0.88 LMNA (0.40) ALDH1A1KDM4E
SCHEMBL6592054 0.86 CYP3A4 (0.30)
SCHEMBL6587765 0.81 LMNA (0.34) ALDH1A1KDM4EMAPTEEDCYP2C9
SCHEMBL6593566 0.76 RXFP1 (0.37) ALDH1A1EEDCYP2C9TSHR
SCHEMBL8432083 0.74 RXFP1 (0.35) ALDH1A1EEDSLC6A2CYP2C9TSHR
SCHEMBL6590388 0.72 SLC6A2 (0.31) SLC6A2
SCHEMBL6589332 0.69 RXFP1 (0.49) ALDH1A1KDM4ECYP2C9TSHR
SCHEMBL6589723 0.67 RXFP1 (0.31) EEDSLC6A2
SCHEMBL6589652 0.65 LMNA (0.33) ALDH1A1EEDCYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0703232-B1 2,3-Dihydro-1H-isoindole derivates, a process for their preparation and their use as serotonin reuptake inhibitors AVENTIS PHARMA INC (US) 2004-06-30 EP claimed
US-5567718-A PSYCHOLOGICAL DISORDERS HOECHST MARION ROUSSEL INC. (US) 1996-10-22 US claimed
EP-0703232-A2 2,3-Dihydro-1H-isoindole derivates, a process for their preparation and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1996-03-27 EP claimed
EP-0703232-B1 2,3-Dihydro-1H-isoindole derivates, a process for their preparation and their use as serotonin reuptake inhibitors AVENTIS PHARMA INC (US) 2004-06-30 EP disclosed
US-5874458-A PSYCHOLOGICAL DISORDERS HOECHST MARION ROUSSEL INC. (US) 1999-02-23 US disclosed
US-5874583-A TREATING DEPRESSION, OBSESSIVE COMPULSIVE DISORDER, STUTTERING, TRICHOTILLOMANIA HOECHST MARION ROUSSEL INC. (US) 1999-02-23 US disclosed
US-5869685-A SEROTONIN REUPTAKE INHIBITORS HOECHST MARION ROUSSEL INC. (US) 1999-02-09 US disclosed
US-5869502-A TREATING DEPRESSION, OBSESSIVE COMPULSIVE DISORDER, STUTTERING, TRICHOTILLOMANIA HOECHST MARION ROUSSEL INC. (US) 1999-02-09 US disclosed
US-5567718-A PSYCHOLOGICAL DISORDERS HOECHST MARION ROUSSEL INC. (US) 1996-10-22 US disclosed
EP-0703232-A2 2,3-Dihydro-1H-isoindole derivates, a process for their preparation and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1996-03-27 EP disclosed