SCHEMBL6589652

SCHEMBL6589652

CC1(C(=CC(=O)O)C(=O)O)c2ccccc2CN1c1ccncc1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.33
BLM P54132 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
EED O75530 1/20 0.32
KDM5A P29375 1/20 0.30
KDM4C Q9H3R0 1/20 0.30
KDM5B Q9UGL1 1/20 0.30
CYP2C9 P11712 2/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HIF1A Q16665 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6589723 0.83 RXFP1 (0.31) RXFP1EED
SCHEMBL8432079 0.83 RXFP1 (0.36) LMNARXFP1EED
SCHEMBL6593270 0.83 RXFP1 (0.36) LMNARXFP1EED
SCHEMBL6590388 0.81 SLC6A2 (0.31)
SCHEMBL6587765 0.71 LMNA (0.34) LMNABLMRXFP1EEDCYP2C9
SCHEMBL6589626 0.68 RXFP1 (0.50) LMNARXFP1EEDCYP2D6TSHR
SCHEMBL8432083 0.68 RXFP1 (0.35) LMNABLMRXFP1EEDCYP2C9
SCHEMBL6593566 0.67 RXFP1 (0.37) LMNARXFP1EEDCYP2C9ALDH1A1
SCHEMBL6592827 0.67 ALDH1A1 (0.33) EEDCYP2C9ALDH1A1CYP2D6TSHR
SCHEMBL6589528 0.65 MMP9 (0.32) EEDCYP2C9ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0703232-B1 2,3-Dihydro-1H-isoindole derivates, a process for their preparation and their use as serotonin reuptake inhibitors AVENTIS PHARMA INC (US) 2004-06-30 EP claimed