SCHEMBL8433460

SCHEMBL8433460

CN(C)CCCC1(OC(=O)/C=C\C(=O)OC2(CCCN(C)C)c3ccccc3CN2c2ccncc2)c2ccccc2CN1c1ccncc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
KDM4E B2RXH2 4/20 0.33
PKM P14618 1/20 0.33
SLC6A4 P31645 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CHRM2 P08172 2/20 0.32
CHRM4 P08173 2/20 0.32
CHRM5 P08912 2/20 0.32
CHRM1 P11229 2/20 0.32
CACNA1B Q00975 1/20 0.31
HSP90B1 P14625 1/20 0.31
TRAP1 Q12931 1/20 0.31
NAMPT P43490 2/20 0.31
CHRM3 P20309 1/20 0.31
ALDH1A1 P00352 1/20 0.30
BCHE P06276 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6589528 0.88 MMP9 (0.32) KDM4EALDH1A1
SCHEMBL6592827 0.85 ALDH1A1 (0.33) KDM4EPKMALDH1A1
SCHEMBL6592054 0.82 CYP3A4 (0.30)
SCHEMBL6587765 0.77 LMNA (0.34) LMNAKDM4ENAMPTALDH1A1
SCHEMBL6593566 0.73 RXFP1 (0.37) LMNAALDH1A1
SCHEMBL8432083 0.71 RXFP1 (0.35) LMNAALDH1A1
SCHEMBL6589332 0.64 RXFP1 (0.49) LMNAKDM4EL3MBTL1ALDH1A1
SCHEMBL6590388 0.63 SLC6A2 (0.31)
Fumaric Acid SCHEMBL8433463 0.63 HRH1 (0.42) LMNAKDM4EL3MBTL1ALDH1A1
Maleic Acid SCHEMBL8433458 0.63 HRH1 (0.42) LMNAKDM4EL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874583-A TREATING DEPRESSION, OBSESSIVE COMPULSIVE DISORDER, STUTTERING, TRICHOTILLOMANIA HOECHST MARION ROUSSEL INC. (US) 1999-02-23 US disclosed