SCHEMBL6589596

SCHEMBL6589596

O=C(O)C(O)(c1ccccc1C1CCN(CCC=C2CCCC2)CC1)C1CCC1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 13/20 0.42
CHRM2 P08172 4/20 0.42
CHRM1 P11229 4/20 0.42
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
RBP4 P02753 2/20 0.39
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6589130 0.86 CHRM3 (0.58) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL6587443 0.80 OPRL1 (0.43) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL6589592 0.77 ALDH1A1 (0.57) CHRM3CHRM2CHRM1HTT
SCHEMBL17871674 0.74 ALDH1A1 (0.52) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL6592856 0.73 CHRM2 (0.74) CHRM3CHRM2CHRM1
Bromomethane SCHEMBL19839345 0.72 ALDH1A1 (0.50) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL6589288 0.72 GPR119 (0.49) RBP4
SCHEMBL6590742 0.71 KEAP1 (0.43) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL4967978 0.69 ALDH1A1 (0.46) CHRM3CHRM2CHRM1KEAP1NFE2L2
SCHEMBL2596487 0.68 KEAP1 (0.50) CHRM3CHRM2CHRM1KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823423-B1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMA CO LTD (JP) 2004-06-16 EP claimed
EP-0823423-B1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMA CO LTD (JP) 2004-06-16 EP disclosed
US-5750540-A SIDE EFFECT REDUCTION BANYU PHARMACEUTICAL CO., LTD. (JP) 1998-05-12 US disclosed
EP-0823423-A1 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1998-02-11 EP disclosed