SCHEMBL6592525

SCHEMBL6592525

CC1CCCCC1.COc1nsnc1N1CCN(C[C@@H](Cc2cccnc2)NC(=O)O)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.72
DRD4 P21917 1/20 0.72
DRD3 P35462 1/20 0.72
NPSR1 Q6W5P4 2/20 0.37
LMNA P02545 2/20 0.37
HSD17B10 Q99714 2/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.36
C3AR1 Q16581 2/20 0.35
CHRM4 P08173 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6177540 0.79 MEN1 (0.46) HTR1ADRD4DRD3NPSR1ALDH1A1
SCHEMBL6586789 0.76 HTR1A (0.61) HTR1ADRD4DRD3HSD17B10ALDH1A1
SCHEMBL6588617 0.73 HTR1A (0.61) HTR1ADRD4DRD3NPSR1LMNA
SCHEMBL6586733 0.73 HTR1A (0.61) HTR1ADRD4DRD3NPSR1LMNA
SCHEMBL6181828 0.69 MEN1 (0.45) HTR1ADRD4NPSR1ALDH1A1MAPT
SCHEMBL6176194 0.69 MEN1 (0.52) HTR1ADRD4NPSR1ALDH1A1GAA
SCHEMBL6588614 0.69 HTR1A (0.66) HTR1ADRD4DRD3NPSR1LMNA
SCHEMBL6586728 0.69 HTR1A (0.66) HTR1ADRD4DRD3NPSR1LMNA
SCHEMBL28746727 0.67 KMT2A (0.49) HTR1ADRD4DRD3LMNAHSD17B10
SCHEMBL7968949 0.66 MEN1 (0.45) HTR1ADRD4DRD3POLBC3AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161424-B1 NEW DIAZOLE DERIVATIVES AS SEROTONERGIC AGENTS WYETH CORP (US) 2004-06-02 EP claimed