SCHEMBL6592979

SCHEMBL6592979

O=Cc1c(Cc2ccccc2)[nH]c2ccccc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 6/20 0.66
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
HPGD P15428 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
TSHR P16473 2/20 0.48
CYP2C19 P33261 2/20 0.48
MTNR1A P48039 2/20 0.48
MTNR1B P49286 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
CYP2C9 P11712 1/20 0.48
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
IMPDH2 P12268 1/20 0.46
MAPT P10636 2/20 0.43
CYP2D6 P10635 1/20 0.42
ALOX15 P16050 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
KIF11 P52732 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28003901 0.87 AHR (0.63) AHRMEN1KMT2AALDH1A1KDM4E
SCHEMBL9300229 0.87 AHR (0.59) AHRMEN1KMT2AHPGDCYP1A2
SCHEMBL8685679 0.87 AHR (0.59) AHRMEN1KMT2AHPGDCYP1A2
SCHEMBL28239180 0.86 AHR (0.52) AHRMEN1KMT2AHPGDMAPT
SCHEMBL28863000 0.85 AHR (0.54) AHRMEN1KMT2AHPGDCYP1A2
SCHEMBL27364002 0.85 AHR (0.49) AHRMEN1KMT2AHPGDCYP1A2
SCHEMBL28735487 0.85 AHR (0.49) AHRMEN1KMT2AHPGDCYP1A2
SCHEMBL28490003 0.83 MAOA (0.51) AHRMEN1KMT2AMAPTSMN1; SMN2
SCHEMBL8804361 0.82 KMT2A (0.48) AHRMEN1KMT2AHPGDCYP1A2
SCHEMBL4323256 0.82 GSK3B (0.51) AHRMEN1KMT2AIMPDH2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110330535-B N-heterocyclic carbene-based mixed nickel (II) complex and application thereof 苏州大学 2022-04-15 CN disclosed
CN-110330535-B N-heterocyclic carbene-based mixed nickel (II) complex and application thereof 苏州大学 2022-04-15 CN disclosed
CN-110330535-A N-heterocyclic carbine base mixed matching nickel (II) complex and its application 苏州大学 2019-10-15 CN disclosed
CN-108358923-A Sophoridine pyrroles, indole derivatives and the preparation method and application thereof 广西大学 2018-08-03 CN disclosed
CN-108047226-A Matrine pyrroles, indole derivatives and preparation method and application 广西大学 2018-05-18 CN disclosed
CN-103172577-B 4-amido quinazoline and 4-aminoquinoline compounds and uses thereof SHENYANG PHARMACEUTICAL UNIVERSITY (CN) 2015-10-07 CN disclosed
CN-102643272-B Novel thieno [3, 2-d] pyrimidine compound UNIV SHENYANG PHARMACEUTICAL 2015-03-11 CN disclosed
CN-103172577-A 4-aminoquinoline and 4-aminoquinoline compound and applications of compound UNIV SHENYANG PHARMACEUTICAL 2013-06-26 CN disclosed
EP-1359915-A4 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM (US) 2004-07-21 EP disclosed
EP-1351687-A4 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2004-01-21 EP disclosed
EP-1359915-A1 UROTENSIN-II RECEPTOR ANTAGONISTS Smithkline Beecham (US) 2003-11-12 EP disclosed
EP-1351687-A2 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2003-10-15 EP disclosed
WO-2002058702-A1 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (GB) 2002-08-01 WO disclosed
WO-2002047456-A2 UROTENSIN-II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2002-06-20 WO disclosed
EP-0837870-A1 SYNTHETIC MODIFICATION TO SPINOSYN COMPOUNDS DOWELANCO (US) 1998-04-29 EP disclosed
WO-1997000265-A1 SYNTHETIC MODIFICATION TO SPINOSYN COMPOUNDS DOWELANCO (US) 1997-01-03 WO disclosed
EP-0375133-A1 Alpha-amino-indole-3-acetic acids useful as anti-diabetic, anti-obesity and anti-atherosclerotic agents THE UPJOHN COMPANY (US) 1990-06-27 EP disclosed