SCHEMBL6594963

SCHEMBL6594963

O=[C]c1c(C(=O)N2CCCC2)[nH]c2cc(Cl)ccc2c1=O

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.57
MAPT P10636 1/20 0.46
HRH4 Q9H3N8 4/20 0.45
HRH3 Q9Y5N1 1/20 0.45
MAP2 P11137 1/20 0.45
ALOX5 P09917 1/20 0.43
MAT2A P31153 2/20 0.43
MDM2 Q00987 1/20 0.41
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
KDM4E B2RXH2 2/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
MAPK1 P28482 1/20 0.39
BLM P54132 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5757658 0.82 PTGS2 (0.58) PTGS2MAPTHRH4HRH3MAP2
SCHEMBL6994667 0.74 HRH4 (0.64) PTGS2HRH4HRH3MAT2ACA12
SCHEMBL10857861 0.72 PTGS2 (0.49) PTGS2MAPTHRH4HRH3MAT2A
SCHEMBL6388357 0.69 ALPL (0.45) PTGS2ALOX5KDM4EHPGDMAPK1
SCHEMBL6384274 0.69 PDE1A (0.51) PTGS2MAPTKDM4EHSD17B10LMNA
SCHEMBL14543827 0.66 PARP1 (0.62) MAT2ACA12CA9KDM4EMEN1
SCHEMBL2730991 0.66 PTGS2 (0.52) PTGS2MAPTMAP2ALOX5KDM4E
SCHEMBL602787 0.65 HRH4 (0.62) PTGS2HRH4HRH3MAP2ALOX5
SCHEMBL24196838 0.63 ALDH1A1 (0.49) PTGS2MAPTHRH4MAP2MEN1
SCHEMBL29586144 0.63 PARP1 (0.58) MAT2ACA12CA9KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244663-B1 COMPOUNDS AND METHODS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2004-08-25 EP disclosed