SCHEMBL6596273

SCHEMBL6596273

O=C(O)c1cc(OCc2ccccc2)c2ccc(C#Cc3ccccc3)c(OCc3ccccc3)c2n1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
XDH P47989 3/20 0.44
MCL1 Q07820 3/20 0.42
PTGER1 P34995 6/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.39
P4HTM Q9NXG6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080107 0.92 ADORA3 (0.39) XDHMCL1PTGER1PTGDR2
SCHEMBL6594101 0.88 MCL1 (0.43) XDHMCL1PTGER1P4HTM
SCHEMBL6598552 0.86 XDH (0.42) XDHMCL1PTGER1P4HTM
SCHEMBL6596521 0.84 XDH (0.40) XDHMCL1PTGER1
SCHEMBL6593178 0.82 XDH (0.47) XDHMCL1PTGER1P4HTM
SCHEMBL6591653 0.81 MRGPRX4 (0.46) XDHMCL1PTGER1
SCHEMBL6592610 0.81 XDH (0.49) XDHMCL1
SCHEMBL6596585 0.81 THRA (0.45) MCL1PTGER1P4HTM
SCHEMBL6592323 0.80 MCL1 (0.48) XDHMCL1PTGER1
SCHEMBL6080093 0.79 MMP2 (0.36) XDHPTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed