SCHEMBL6601729

SCHEMBL6601729

O=C(O)[C@]1(F)C=C[C@H](c2ccccc2)C=C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.35
HTR2C P28335 2/20 0.35
HTR2B P41595 2/20 0.35
EDNRA P25101 1/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
HDAC4 P56524 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
CA2 P00918 1/20 0.32
EPHX1 P07099 1/20 0.32
OPRK1 P41145 1/20 0.31
AKR1C3 P42330 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2508140 1.00 HTR2A (0.35) HTR2AHTR2CHTR2BEDNRAMEN1
SCHEMBL316145 0.80 EDNRA (0.35) EDNRAMAPK1CYP2C19HDAC4HDAC3
SCHEMBL1119643 0.78 THRB (0.35) EDNRAMAPK1CYP2C19HDAC4HDAC3
SCHEMBL746904 0.78 HTR2A (0.38) HTR2AHTR2CHTR2BCA2RECQL
SCHEMBL1577842 0.77 HTR2A (0.41) HTR2AHTR2CHTR2BMEN1KMT2A
SCHEMBL3583056 0.77 GRM1 (0.35) EDNRAMEN1KMT2ALMNAMAPK1
SCHEMBL2121106 0.77 KDM1A (0.34) EDNRAMAPK1CYP2C19HDAC4HDAC3
SCHEMBL4371618 0.77 SLC9A1 (0.36) EDNRAMAPK1CYP2C19OPRK1POLB
SCHEMBL16290377 0.77 HSD11B1 (0.38) HTR2AHTR2CHTR2BEDNRAMEN1
SCHEMBL6709305 0.77 EDNRA (0.34) EDNRAMAPK1CYP2C19HDAC4HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1432693-A2 MCH RECEPTOR ANTAGONISTS Taisho Pharmaceutical Co. Ltd. (JP) 2004-06-30 EP disclosed
WO-2003028641-A2 MCH RECEPTOR ANTAGONISTS TAISHO PHARMACEUTICAL CO., LTD. (JP) 2003-04-10 WO disclosed