SCHEMBL6605626

SCHEMBL6605626

COc1ccc(C2SC(=O)NC2=O)cc1C(=O)NCc1cccc(C(F)(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 11/20 0.56
ROCK2 O75116 1/20 0.49
ROCK1 Q13464 1/20 0.49
LMNA P02545 2/20 0.47
PPARD Q03181 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KCNQ3 O43525 1/20 0.46
KCNQ2 O43526 1/20 0.46
PSEN1 P49768 3/20 0.46
PSEN2 P49810 3/20 0.46
APH1B Q8WW43 3/20 0.46
NCSTN Q92542 3/20 0.46
APH1A Q96BI3 3/20 0.46
PSENEN Q9NZ42 3/20 0.46
HPGD P15428 1/20 0.46
PPARG P37231 3/20 0.45
MLYCD O95822 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6607449 0.90 PPARA (0.58) PPARAPPARDPSEN1PSEN2APH1B
SCHEMBL6239522 0.85 PPARA (0.59) PPARAROCK2ROCK1LMNAPPARD
SCHEMBL27360910 0.81 PPARA (0.47) PPARAPPARDPSEN1PSEN2APH1B
SCHEMBL27388283 0.81 PPARA (0.48) PPARAPPARDPSEN1PSEN2APH1B
SCHEMBL27529292 0.80 PPARA (0.49) PPARAPPARDPSEN1PSEN2APH1B
SCHEMBL20125593 0.75 PPARA (0.61) PPARAPPARDPSEN1PSEN2APH1B
SCHEMBL3922 0.75 PPARA (0.61) PPARAPPARDPSEN1PSEN2APH1B
SCHEMBL14379043 0.75 PPARA (0.61) PPARAPPARDPSEN1PSEN2APH1B
SCHEMBL29358494 0.75 PPARA (0.61) PPARAPPARDPSEN1PSEN2APH1B
SCHEMBL6236525 0.73 ROCK2 (0.49) PPARAROCK2ROCK1LMNAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0881219-B1 N-SUBSTITUTED DIOXOTHIAZOLIDYLBENZAMIDE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2004-04-07 EP claimed
CN-1065863-C N-substituted dioxothiazolidylbenzamide derivatives and process for producing the same KYORIN SEIYAKU KK (JP) 2001-05-16 CN claimed
US-5948803-A IMPROVE THE INSULIN RESISTANCE AND HAVE POTENT HYPOGLYCEMIC EFFECT AND LIPID-LOWERING EFFECT KYORIN PHARMACEUTICAL CO., LTD. (JP) 1999-09-07 US claimed
CN-1205695-A N-substituted dioxothiazolidylbenzamide derivatives and process for producing the same KYORIN SEIYAKU KK (JP) 1999-01-20 CN claimed
EP-0881219-A1 N-SUBSTITUTED DIOXOTHIAZOLIDYLBENZAMIDE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1998-12-02 EP claimed
JP-9169746-A None JP disclosed
JP-H09169746-A N-SUBSTITUTED DIOXOTHIAZOLIDYLBENZAMIDE DERIVATIVE AND ITS PRODUCTION KYORIN PHARMACEUT CO LTD 1997-06-30 JP disclosed