SCHEMBL6607386

SCHEMBL6607386

CON(Cc1ccccc1)S(=O)(=O)c1ccc(CC(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 12/20 0.50
PTGES O14684 3/20 0.50
CXCR3 P49682 2/20 0.50
TAS2R8 Q9NYW2 1/20 0.50
AKR1B1 P15121 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
NR3C1 P04150 1/20 0.46
ALOX5 P09917 1/20 0.46
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5450808 0.81 ALDH1A1 (0.62) AKR1B1MEN1KMT2AMAPT
SCHEMBL1279080 0.80 TAS2R14 (0.77) TAS2R14PTGESCXCR3TAS2R8
SCHEMBL5448485 0.79 TAS2R14 (0.61) TAS2R14CXCR3MEN1KMT2APOLB
SCHEMBL6609506 0.79 HTT (0.66) TAS2R14AKR1B1MEN1KMT2A
SCHEMBL5459206 0.79 PTGES (0.46) TAS2R14PTGESCXCR3TAS2R8AKR1B1
SCHEMBL2514583 0.74 ALDH1A1 (0.54) PTGESAKR1B1ALOX5MAPT
SCHEMBL5452529 0.71 LMNA (0.59) TAS2R14MEN1KMT2A
Phenylacetic Acid SCHEMBL29521265 0.71 AKR1B1 (0.94) AKR1B1MEN1KMT2APOLB
SCHEMBL5459724 0.70 ALDH1A1 (0.46) TAS2R14PTGESAKR1B1KMT2AALOX5
Phenylacetic Acid SCHEMBL23925805 0.69 AKR1B1 (0.74) AKR1B1MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451172-A1 THERAPEUTIC ISOQUINOLINE COMPOUNDS AstraZeneca AB (SE) 2004-09-01 EP disclosed
WO-2003037887-A1 THERAPEUTIC ISOQUINOLINE COMPOUNDS ASTRAZENECA AB (SE) 2003-05-08 WO disclosed