Benzamide

Benzamide

SCHEMBL6607765

NC(=O)c1ccccc1.c1c[nH]c(N2CCNCC2)c1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 2/20 0.50
TSHR P16473 2/20 0.49
HSD17B10 Q99714 2/20 0.49
USP2 O75604 1/20 0.49
ALDH1A1 P00352 1/20 0.49
SIGMAR1 Q99720 2/20 0.46
POLB P06746 1/20 0.46
CYP3A4 P08684 1/20 0.46
PARP1 P09874 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C19 P33261 1/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46
PMP22 Q01453 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
SLC6A4 P31645 1/20 0.43
PRKD1 Q15139 3/20 0.42
PRKD2 Q9BZL6 3/20 0.42
HTR6 P50406 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4491073 0.81 ADRB1 (0.48) ALDH1A1SIGMAR1CYP3A4CYP2C19SLC6A4
Phenylpiperazine SCHEMBL29235064 0.80 TSHR (0.69) OPRD1TSHRHSD17B10USP2ALDH1A1
Benzamide SCHEMBL28329540 0.76 HRH4 (0.50) OPRD1TSHRHSD17B10USP2ALDH1A1
Benzamide SCHEMBL572737 0.76 TSHR (0.73) OPRD1TSHRHSD17B10USP2ALDH1A1
Benzamide SCHEMBL1472873 0.75 OPRD1 (0.57) OPRD1TSHRHSD17B10USP2ALDH1A1
Benzamide SCHEMBL4726018 0.72 TSHR (0.67) OPRD1TSHRHSD17B10USP2ALDH1A1
Benzamide SCHEMBL1474746 0.72 SIGMAR1 (0.58) OPRD1TSHRHSD17B10USP2ALDH1A1
SCHEMBL572738 0.72 ACVR1 (0.66) OPRD1TSHRHSD17B10USP2ALDH1A1
Benzamide SCHEMBL1220629 0.71 DRD2 (0.68) OPRD1TSHRHSD17B10USP2ALDH1A1
Benzamide SCHEMBL694831 0.71 TSHR (0.64) OPRD1TSHRHSD17B10USP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451172-A1 THERAPEUTIC ISOQUINOLINE COMPOUNDS AstraZeneca AB (SE) 2004-09-01 EP disclosed
WO-2003037887-A1 THERAPEUTIC ISOQUINOLINE COMPOUNDS ASTRAZENECA AB (SE) 2003-05-08 WO disclosed