SCHEMBL6608637

SCHEMBL6608637

C=CC[Si](CC=C)(CC=C)N(C(N)=O)[Si](CC=C)(CC=C)CC=C

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
FGFR4 P22455 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9449766 0.76 ALDH1A1 (0.33) ALDH1A1
SCHEMBL4854523 0.71
SCHEMBL2537847 0.70 TSHR (0.30) TSHR
SCHEMBL7591793 0.68 ALDH1A1 (0.35) ALDH1A1TSHRFGFR4
SCHEMBL8060637 0.67
SCHEMBL8775960 0.67 ALOX15 (0.32)
SCHEMBL6267318 0.65 LMNA (0.39) ALDH1A1
SCHEMBL7592451 0.64
SCHEMBL3801722 0.63 ALDH1A1 (0.35) ALDH1A1TSHRFGFR4
SCHEMBL9328869 0.62 ALDH1A1 (0.33) ALDH1A1TSHRFGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0842927-B1 3-Amido-chromanylsulfonyl(thio)ureas, process for their preparation, their use and medicaments containing them AVENTIS PHARMA GMBH (DE) 2004-02-25 EP claimed
EP-0729954-B1 Substituted thiophene sulfonyl ureas and thioureas, process for their preparation, their use as medicaments HOECHST AG (DE) 2003-09-03 EP claimed
US-6506937-B2 Used as antiarrhythmics SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2003-01-14 US claimed
EP-0726250-B1 Substituted benzenesulfonylureas and -thioureas, process for their preparation and their use in the production of pharmaceutical preparations as well as pharmaceutical preparations containing them HOECHST AG (DE) 2000-11-02 EP claimed
EP-0779288-B1 Substituted chromanylsulfonyl(thio)ureas, process for their preparation, their use in pharmaceutical compositions and preparations containing them HOECHST AG (DE) 2000-03-29 EP claimed
EP-0727416-B1 Substituted benzenesulfonylureas and -thioureas, process for their preparation, their use as medicament or diagnostic agent, as well as medicaments containing them HOECHST AG (DE) 2000-01-26 EP claimed
US-5849755-A 3-amidochromanylsulfonyl(thio)ureas, processes for their preparation, their use, and pharmaceutical preparations comprising them HOECHST AKTIENGESELLSCHAFT (DE) 1998-12-15 US claimed
US-5811448-A PHARMACEUTICALS USEFUL FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS HOECHST AKTIENGESELLSCHAFT (DE) 1998-09-22 US claimed
EP-0830362-A4 PROCESS FOR THE SYNTHESIS OF VINYL SULFENIC ACID DERIVATIVES LILLY CO ELI (US) 1998-09-02 EP claimed
US-5792788-A FOR TREATMENT OF CARDIAC DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1998-08-11 US claimed
EP-0830362-A1 PROCESS FOR THE SYNTHESIS OF VINYL SULFENIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1998-03-25 EP claimed
US-5652268-A TREATING CARDIOVASCULAR DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-07-29 US claimed
WO-1996040693-A1 PROCESS FOR THE SYNTHESIS OF VINYL SULFENIC ACID DERIVATIVES ELI LILLY AND COMPANY (US) 1996-12-19 WO claimed
US-5512701-A REACTING SULFOXIDE DERIVATIVE WITH A SILYATING AGENT TO FORM SULFENATE SILYL ESTER, OPTIONALLY REACTING INTERMEDIATE WITH AN AMINE AND/OR A MERCAPTAN ELI LILLY AND COMPANY (US) 1996-04-30 US claimed
US-10358526-B2 Moisture-curing polyether carbonate containing alkoxysilyl groups COVESTRO DEUTSCHLAND AG (DE) 2019-07-23 US disclosed
US-20170313816-A1 MOISTURE-CURING POLYETHER CARBONATE CONTAINING ALKOXYSILYL GROUPS COVESTRO DEUTSCHLAND AG (DE) 2017-11-02 US disclosed
US-6506937-B2 Used as antiarrhythmics SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2003-01-14 US disclosed
EP-0024292-B1 PROCESS FOR THE SEPARATION OF URSODEOXYCHOLIC ACID FROM CHENODEOXYCHOLIC ACID AND PRODUCTS OBTAINED DURING THE PROCESS BLASCHIM S.p.A. (IT) 1983-06-01 EP disclosed
US-4316848-A Process for the purification of ursodeoxycholic acid BLASINACHIM S.P.A (IT) 1982-02-23 US disclosed
EP-0024292-A1 Process for the separation of ursodeoxycholic acid from chenodeoxycholic acid and products obtained during the process BLASCHIM S.p.A. (IT) 1981-03-04 EP disclosed